SCHEMBL28346142

SCHEMBL28346142

CCOC(=O)C1=C(C)NC(C=O)NC1c1ccc(Br)cc1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HSD17B10 Q99714 1/20 0.45
DHFR P00374 1/20 0.44
CA12 O43570 2/20 0.43
CA1 P00915 2/20 0.43
CA2 P00918 2/20 0.43
CA7 P43166 2/20 0.43
CA9 Q16790 2/20 0.43
ALDH1A1 P00352 3/20 0.42
MAPT P10636 2/20 0.42
LMNA P02545 1/20 0.42
HTT P42858 1/20 0.42
POLB P06746 1/20 0.42
L3MBTL1 Q9Y468 1/20 0.42
KDM4E B2RXH2 1/20 0.40
TSHR P16473 1/20 0.40
SMN1; SMN2 Q16637 1/20 0.40
GAA P10253 2/20 0.40
MEN1 O00255 1/20 0.40
KMT2A Q03164 1/20 0.40
GUSB P08236 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28345988 0.88 MEN1 (0.49) HSD17B10DHFRCA12CA1CA2
SCHEMBL28346144 0.88 ABCC1 (0.54) HSD17B10CA12CA1CA2CA7
SCHEMBL28349893 0.88 SMN1; SMN2 (0.46) MAPTLMNASMN1; SMN2GAAMEN1
SCHEMBL28881024 0.86 KIF11 (0.48) DHFRALDH1A1MAPTLMNAHTT
SCHEMBL28345331 0.79 MAPK1 (0.51) DHFRALDH1A1MAPTLMNAHTT
SCHEMBL28342583 0.76 TSHR (0.63) HSD17B10DHFRCA1CA2ALDH1A1
SCHEMBL28490632 0.76 HSD17B10 (0.73) HSD17B10CA12CA1CA2CA7
SCHEMBL27766887 0.76 HSD17B10 (0.38) HSD17B10DHFRCA12CA1CA2
SCHEMBL28350092 0.75 ALDH1A1 (0.48) HSD17B10CA1CA2ALDH1A1MAPT
SCHEMBL28562281 0.75 DHFR (0.77) DHFRCA12CA1CA2CA7

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-108129398-B Synthesis method of 4-halogenated phenyl-5-ethoxycarbonyl-6-methyl-3, 4-dihydropyrimidine-2 (1H) -ketone 大连大学 2020-01-17 CN disclosed