SCHEMBL28884135

SCHEMBL28884135

CCC(C)Nc1nc(N)nc(-c2ccccc2)n1

nearest known ligand 0.56

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
NPSR1 Q6W5P4 1/20 0.56
ADORA2A P29274 2/20 0.51
ADORA1 P30542 2/20 0.51
POLB P06746 1/20 0.51
ADORA3 P0DMS8 1/20 0.51
ADORA2B P29275 1/20 0.51
TPH1 P17752 10/20 0.51
HSP90AA1 P07900 1/20 0.45
HSP90AB1 P08238 1/20 0.45
GPR68 Q15743 3/20 0.44
HTR1A P08908 1/20 0.44
HRH4 Q9H3N8 1/20 0.43
ALDH1A1 P00352 1/20 0.41
NPC1 O15118 1/20 0.41
TSHR P16473 1/20 0.41
HSD17B10 Q99714 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16370342 0.89 ALDH1A1 (0.49) ADORA2AADORA1ADORA3HSP90AA1ALDH1A1
SCHEMBL28184778 0.84 ADORA2A (0.58) NPSR1ADORA2AADORA1POLBADORA3
SCHEMBL11425373 0.80 NPSR1 (0.54) NPSR1ADORA2AADORA1POLBADORA3
SCHEMBL10059800 0.79 L3MBTL1 (0.47) HSP90AA1ALDH1A1TSHRHSD17B10
SCHEMBL6269189 0.78 NPSR1 (0.71) NPSR1ADORA2AADORA1POLBADORA3
SCHEMBL9112534 0.78 NPSR1 (0.51) NPSR1ADORA2AADORA1POLBADORA3
SCHEMBL5159281 0.78 NPSR1 (0.54) NPSR1ADORA2AADORA1POLBADORA3
SCHEMBL11164961 0.77 NPSR1 (0.50) NPSR1ADORA2AADORA1POLBADORA3
SCHEMBL29560835 0.77 IDH2 (0.52) NPC1TSHRHSD17B10
SCHEMBL15102522 0.77 IDH2 (0.52) NPC1TSHRHSD17B10

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-105473560-B Therapeutically active compounds and methods of use thereof 安吉奥斯医药品有限公司 2020-01-17 CN claimed
CN-111087353-B Therapeutically active compounds and methods of use thereof 法国施维雅药厂 2023-10-24 CN disclosed
CN-111087353-A Therapeutically active compounds and methods of use thereof 安吉奥斯医药品有限公司 2020-05-01 CN disclosed
CN-105473560-B Therapeutically active compounds and methods of use thereof 安吉奥斯医药品有限公司 2020-01-17 CN disclosed