SCHEMBL28889276

SCHEMBL28889276

Cc1ccnc(C(C#N)c2ccccc2Cl)c1

nearest known ligand 0.54

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 4/20 0.54
OPRM1 P35372 3/20 0.42
OPRL1 P41146 3/20 0.42
CTSA P10619 1/20 0.41
GAA P10253 3/20 0.40
L3MBTL1 Q9Y468 1/20 0.40
MDM2 Q00987 1/20 0.38
SLC6A2 P23975 1/20 0.37
SLC6A4 P31645 1/20 0.37
SLC6A3 Q01959 1/20 0.37
LMNA P02545 1/20 0.36
POLB P06746 1/20 0.36
CYP2C19 P33261 1/20 0.36
MAPK9 P45984 1/20 0.34
MAPK10 P53779 1/20 0.34
MAPT P10636 2/20 0.34
CYP19A1 P11511 1/20 0.34
MEN1 O00255 1/20 0.34
NPC1 O15118 1/20 0.34
HPGD P15428 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28889180 0.81 ALDH1A1 (0.51) ALDH1A1GAAL3MBTL1LMNAPOLB
SCHEMBL11631926 0.80 ALDH1A1 (0.60) ALDH1A1OPRM1OPRL1GAAL3MBTL1
SCHEMBL28889203 0.80 ALDH1A1 (0.50) ALDH1A1GAAL3MBTL1LMNAPOLB
SCHEMBL28889217 0.80 ALDH1A1 (0.50) ALDH1A1OPRM1OPRL1GAALMNA
SCHEMBL9664891 0.74 ALDH1A1 (0.62) ALDH1A1OPRL1GAAL3MBTL1SLC6A2
SCHEMBL6767570 0.73 ALDH1A1 (0.55) ALDH1A1OPRM1OPRL1GAALMNA
SCHEMBL28889227 0.72 CTSA (0.47) OPRM1OPRL1CTSAMDM2SLC6A2
SCHEMBL5655425 0.71 ALDH1A1 (0.48) ALDH1A1GAAL3MBTL1LMNAMAPT
SCHEMBL15034193 0.70 UHRF1 (0.43) ALDH1A1GAAL3MBTL1SLC6A2SLC6A4
SCHEMBL29031386 0.69 ALDH1A1 (0.40) ALDH1A1OPRM1OPRL1GAAL3MBTL1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2022222911-A1 PYRIMIDONE COMPOUND AND USE THEREOF 武汉人福创新药物研发中心有限公司 2022-10-27 WO disclosed
CN-115215862-A Pyrimidone compounds and uses thereof 武汉人福创新药物研发中心有限公司 2022-10-21 CN disclosed