SCHEMBL28889227

SCHEMBL28889227

Cc1ccnc(C(C(N)=O)c2ccccc2Cl)c1

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CTSA P10619 4/20 0.47
OPRM1 P35372 4/20 0.41
OPRL1 P41146 4/20 0.41
NPC1 O15118 2/20 0.40
RAB9A P51151 2/20 0.40
SMN1; SMN2 Q16637 2/20 0.40
MEN1 O00255 1/20 0.40
MAPT P10636 1/20 0.40
HPGD P15428 1/20 0.40
NFKB1 P19838 1/20 0.40
NFKB2 Q00653 1/20 0.40
KMT2A Q03164 1/20 0.40
RELA Q04206 1/20 0.40
MDM2 Q00987 1/20 0.39
CRHR1 P34998 1/20 0.37
CXCL8 P10145 1/20 0.36
PKM P14618 1/20 0.36
CDK5 Q00535 1/20 0.36
KLF5 Q13887 1/20 0.36
CDK5R1 Q15078 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28889260 0.82 SMARCA2 (0.38) CTSAOPRM1OPRL1SMN1; SMN2CXCL8
SCHEMBL28889221 0.81 ADRB2 (0.41) OPRL1MEN1MAPTHPGDKMT2A
SCHEMBL28889189 0.80 CTSA (0.45) CTSAOPRM1OPRL1NPC1RAB9A
SCHEMBL28889272 0.80 OPRL1 (0.38) OPRM1OPRL1
SCHEMBL28889168 0.78 CTSA (0.43) CTSAOPRM1OPRL1NPC1RAB9A
SCHEMBL28889346 0.77 CTSA (0.42) CTSAOPRM1OPRL1NPC1RAB9A
SCHEMBL28889276 0.72 ALDH1A1 (0.54) CTSAOPRM1OPRL1NPC1RAB9A
SCHEMBL19716970 0.71 PLAU (0.43) NPC1RAB9ASMN1; SMN2MEN1MAPT
SCHEMBL28889339 0.71 ADRB2 (0.42) CTSA
SCHEMBL29718864 0.70 ACP3 (0.50) MEN1KMT2ACXCL8

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2022222911-A1 PYRIMIDONE COMPOUND AND USE THEREOF 武汉人福创新药物研发中心有限公司 2022-10-27 WO disclosed
CN-115215862-A Pyrimidone compounds and uses thereof 武汉人福创新药物研发中心有限公司 2022-10-21 CN disclosed