SCHEMBL28889288

SCHEMBL28889288

NC(=O)C(c1cc(C(F)(F)F)ccn1)c1ncccc1Cl

nearest known ligand 0.54

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MEN1 O00255 2/20 0.39
KMT2A Q03164 2/20 0.39
KDM4E B2RXH2 1/20 0.39
HSP90AA1 P07900 1/20 0.39
MAPT P10636 1/20 0.39
NPSR1 Q6W5P4 1/20 0.39
L3MBTL1 Q9Y468 1/20 0.39
ADRB2 P07550 1/20 0.38
P2RX7 Q99572 2/20 0.38
KCNH2 Q12809 2/20 0.38
S1PR1 P21453 1/20 0.38
S1PR3 Q99500 1/20 0.38
PRKDC P78527 1/20 0.38
NOS3 P29474 1/20 0.37
NOS2 P35228 1/20 0.37
TRPV1 Q8NER1 2/20 0.37
TRPA1 O75762 1/20 0.37
KCNN4 O15554 1/20 0.37
ALDH1A1 P00352 1/20 0.37
EPAS1 Q99814 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29893638 1.00 MEN1 (0.39) MEN1KMT2AKDM4EHSP90AA1MAPT
SCHEMBL28889221 0.84 ADRB2 (0.41) MEN1KMT2AKDM4EHSP90AA1MAPT
SCHEMBL28889298 0.81 ADRB2 (0.39) MEN1KMT2AL3MBTL1ADRB2KCNH2
SCHEMBL28959207 0.81 KMT2A (0.40) MEN1KMT2AKDM4EHSP90AA1MAPT
SCHEMBL28889351 0.79 ADRB2 (0.40) KDM4EADRB2NOS3NOS2NR3C2
SCHEMBL24110333 0.78 TACR1 (0.45) ADRB2NOS3NOS2ALDH1A1
SCHEMBL28889283 0.78 ADRB2 (0.41) L3MBTL1ADRB2NOS3NOS2TRPV1
SCHEMBL29893620 0.78 AURKA (0.40) ADRB2NOS3NOS2NR3C2
SCHEMBL28889316 0.78 AURKA (0.40) ADRB2NOS3NOS2NR3C2
SCHEMBL28959168 0.78 HDAC4 (0.44) ADRB2NOS3NOS2NR3C2TRPV3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-115215862-A Pyrimidone compounds and uses thereof 武汉人福创新药物研发中心有限公司 2022-10-21 CN disclosed