SCHEMBL28889221

SCHEMBL28889221

NC(=O)C(c1cc(C(F)(F)F)ccn1)c1ccccc1Cl

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ADRB2 P07550 1/20 0.41
OPRL1 P41146 1/20 0.39
EPAS1 Q99814 1/20 0.38
NOS3 P29474 1/20 0.38
NOS2 P35228 1/20 0.38
MEN1 O00255 2/20 0.38
KMT2A Q03164 2/20 0.38
ALDH1A1 P00352 1/20 0.38
GLA P06280 1/20 0.37
HPGD P15428 1/20 0.37
TP53 P04637 1/20 0.37
KDM4C Q9H3R0 1/20 0.37
RORC P51449 2/20 0.36
RORB Q92753 2/20 0.36
KDR P35968 1/20 0.36
NR3C2 P08235 1/20 0.36
TRPV3 Q8NET8 1/20 0.35
MAPT P10636 2/20 0.35
NPSR1 Q6W5P4 2/20 0.35
KDM4E B2RXH2 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28959168 0.86 HDAC4 (0.44) ADRB2NOS3NOS2NR3C2TRPV3
SCHEMBL28889339 0.86 ADRB2 (0.42) ADRB2NOS3NOS2ALDH1A1NR3C2
SCHEMBL28889367 0.85 ADRB2 (0.41) ADRB2NOS3NOS2ALDH1A1NR3C2
SCHEMBL28889288 0.84 MEN1 (0.39) ADRB2EPAS1NOS3NOS2MEN1
SCHEMBL29893638 0.84 MEN1 (0.39) ADRB2EPAS1NOS3NOS2MEN1
SCHEMBL28994016 0.83 ADRB2 (0.40) ADRB2RORBTRPV3MAPTKDM4E
SCHEMBL28889298 0.82 ADRB2 (0.39) ADRB2NOS3NOS2MEN1KMT2A
SCHEMBL24110333 0.82 TACR1 (0.45) ADRB2NOS3NOS2ALDH1A1
SCHEMBL28889231 0.81 GLA (0.39) OPRL1MEN1KMT2AALDH1A1GLA
SCHEMBL28889307 0.81 ADRB2 (0.38) ADRB2NOS3NOS2ALDH1A1NR3C2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-115867541-A Aminopyrimidinone derivatives 豪夫迈·罗氏有限公司 2023-03-28 CN disclosed
WO-2022222911-A1 PYRIMIDONE COMPOUND AND USE THEREOF 武汉人福创新药物研发中心有限公司 2022-10-27 WO disclosed
CN-115215862-A Pyrimidone compounds and uses thereof 武汉人福创新药物研发中心有限公司 2022-10-21 CN disclosed