SCHEMBL28889331

SCHEMBL28889331

Cc1ccc(C(C(N)=O)c2cc(C(F)(F)F)ccn2)cc1

nearest known ligand 0.43

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
ADRB2 P07550 1/20 0.43
NOS3 P29474 1/20 0.40
NOS2 P35228 1/20 0.40
ALDH1A1 P00352 1/20 0.38
GAA P10253 1/20 0.38
L3MBTL1 Q9Y468 1/20 0.38
NR3C2 P08235 2/20 0.38
AURKA O14965 1/20 0.38
ACACB O00763 1/20 0.36
SORT1 Q99523 2/20 0.36
KEAP1 Q14145 1/20 0.36
NFE2L2 Q16236 1/20 0.36
MAPT P10636 1/20 0.35
AKR1C3 P42330 1/20 0.34
AKR1C2 P52895 1/20 0.34
EPHX1 P07099 1/20 0.34
HRH4 Q9H3N8 1/20 0.34
MEN1 O00255 1/20 0.34
KMT2A Q03164 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL24110333 0.86 TACR1 (0.45) ADRB2NOS3NOS2ALDH1A1AURKA
SCHEMBL29893797 0.86 AURKA (0.42) ADRB2NOS3NOS2ALDH1A1L3MBTL1
SCHEMBL28889226 0.86 AURKA (0.42) ADRB2NOS3NOS2ALDH1A1L3MBTL1
SCHEMBL28889143 0.86 ADRB2 (0.42) ADRB2NOS3NOS2ALDH1A1GAA
SCHEMBL28889273 0.82 ADRB2 (0.40) ADRB2NOS3NOS2ALDH1A1GAA
SCHEMBL28889213 0.81 ADRB2 (0.41) ADRB2ALDH1A1GAAL3MBTL1ACACB
SCHEMBL28889339 0.81 ADRB2 (0.42) ADRB2NOS3NOS2ALDH1A1GAA
SCHEMBL28889325 0.81 ADRB2 (0.42) ADRB2NOS3NOS2ALDH1A1GAA
SCHEMBL30637658 0.80 S1PR1 (0.41) ALDH1A1NR3C2ACACBMAPTMEN1
SCHEMBL24110332 0.80 KCNA5 (0.43) ADRB2AURKASORT1MEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2022222911-A1 PYRIMIDONE COMPOUND AND USE THEREOF 武汉人福创新药物研发中心有限公司 2022-10-27 WO disclosed
CN-115215862-A Pyrimidone compounds and uses thereof 武汉人福创新药物研发中心有限公司 2022-10-21 CN disclosed