SCHEMBL28889273

SCHEMBL28889273

NC(=O)C(c1ccnc(F)c1)c1cc(C(F)(F)F)ccn1

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ADRB2 P07550 1/20 0.40
NOS3 P29474 1/20 0.40
NOS2 P35228 1/20 0.40
AURKA O14965 1/20 0.35
NR3C2 P08235 2/20 0.34
KDM4E B2RXH2 1/20 0.34
EPHX1 P07099 2/20 0.33
SYK P43405 1/20 0.33
KMT2A Q03164 1/20 0.33
ALDH1A1 P00352 1/20 0.33
GAA P10253 1/20 0.33
L3MBTL1 Q9Y468 1/20 0.33
FPR2 P25090 1/20 0.32
SCN9A Q15858 1/20 0.32
KCNN4 O15554 1/20 0.32
SCN10A Q9Y5Y9 1/20 0.32
TRPV3 Q8NET8 1/20 0.32
MAPK1 P28482 1/20 0.32
KMO O15229 1/20 0.32
S1PR1 P21453 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28889143 0.86 ADRB2 (0.42) ADRB2NOS3NOS2AURKANR3C2
SCHEMBL28889170 0.85 HDAC4 (0.43) ADRB2NOS3NOS2AURKANR3C2
SCHEMBL29893770 0.85 HDAC4 (0.43) ADRB2NOS3NOS2AURKANR3C2
SCHEMBL24110333 0.84 TACR1 (0.45) ADRB2NOS3NOS2AURKAEPHX1
SCHEMBL28889331 0.82 ADRB2 (0.43) ADRB2NOS3NOS2AURKANR3C2
SCHEMBL28889226 0.81 AURKA (0.42) ADRB2NOS3NOS2AURKANR3C2
SCHEMBL28889280 0.81 AURKA (0.40) ADRB2NOS3NOS2AURKANR3C2
SCHEMBL29893620 0.81 AURKA (0.40) ADRB2NOS3NOS2AURKANR3C2
SCHEMBL29893670 0.81 AURKA (0.40) ADRB2NOS3NOS2AURKANR3C2
SCHEMBL28889316 0.81 AURKA (0.40) ADRB2NOS3NOS2AURKANR3C2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2022222911-A1 PYRIMIDONE COMPOUND AND USE THEREOF 武汉人福创新药物研发中心有限公司 2022-10-27 WO disclosed
CN-115215862-A Pyrimidone compounds and uses thereof 武汉人福创新药物研发中心有限公司 2022-10-21 CN disclosed