SCHEMBL28889808

SCHEMBL28889808

CC(C)(C)N1CCC(OC(N)=O)(c2ccccc2)CC1

nearest known ligand 0.58

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
OPRM1 P35372 10/20 0.58
KCNH2 Q12809 2/20 0.58
GRIN2D O15399 1/20 0.58
GRIN3B O60391 1/20 0.58
CHRM2 P08172 1/20 0.58
CHRM1 P11229 1/20 0.58
GRIN1 Q05586 1/20 0.58
GRIN2A Q12879 1/20 0.58
GRIN2B Q13224 1/20 0.58
GRIN2C Q14957 1/20 0.58
GRIN3A Q8TCU5 1/20 0.58
OPRK1 P41145 8/20 0.43
OPRD1 P41143 7/20 0.43
DRD3 P35462 1/20 0.41
ALDH1A1 P00352 1/20 0.41
OPRL1 P41146 3/20 0.38
HRH3 Q9Y5N1 1/20 0.37
HSD11B1 P28845 1/20 0.36
SCD5 Q86SK9 1/20 0.36
RORC P51449 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2572169 0.81 AKR1C1 (0.42) OPRM1OPRK1OPRD1DRD3OPRL1
SCHEMBL14164046 0.79 OPRM1 (0.60) OPRM1KCNH2GRIN2DGRIN3BCHRM2
SCHEMBL17465640 0.79 OPRM1 (0.64) OPRM1KCNH2GRIN2DGRIN3BCHRM2
SCHEMBL11289324 0.78 AKR1C1 (0.48) OPRM1OPRK1OPRD1HSD11B1
SCHEMBL26135641 0.78 AKR1C1 (0.44) OPRM1OPRK1OPRD1DRD3HSD11B1
SCHEMBL16418420 0.78 OPRM1 (0.63) OPRM1KCNH2GRIN2DGRIN3BCHRM2
SCHEMBL11275197 0.77 AKR1C1 (0.47) HSD11B1
SCHEMBL5698830 0.76 OPRL1 (0.56) OPRM1CHRM2ALDH1A1OPRL1
SCHEMBL10131784 0.75 OPRM1 (0.61) OPRM1KCNH2GRIN2DGRIN3BCHRM2
Budipine SCHEMBL120041 0.74 OPRM1 (1.00) OPRM1KCNH2GRIN2DGRIN3BCHRM2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-115340545-A Bicyclic heteroaryl derivative and preparation method and application thereof 浙江海正药业股份有限公司 2022-11-15 CN disclosed