SCHEMBL2888992

SCHEMBL2888992

C=CCCCCC[C@H](NC(=O)OCC(C)(C)CC=C)C(=O)N1C[C@H](Oc2cc(-c3ccccc3)nc3cc(OC)c(C=C)cc23)C[C@H]1C(=O)N[C@]1(C(=O)O)C[C@H]1C=C

nearest known ligand 0.44

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
CTSB P07858 1/20 0.44
PPP3CB P16298 1/20 0.44
CYP3A4 P08684 2/20 0.37
ABCC1 P33527 1/20 0.31
ABCC2 Q92887 1/20 0.31
ABCG2 Q9UNQ0 1/20 0.31
AAK1 Q2M2I8 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2889001 1.00 CTSB (0.44) CTSBPPP3CBCYP3A4ABCC1ABCC2
SCHEMBL13026234 0.95 CTSB (0.40) CTSBPPP3CBCYP3A4
SCHEMBL2894812 0.91 AAK1 (0.34) CTSBPPP3CBAAK1
SCHEMBL8221244 0.91 AAK1 (0.34) CTSBPPP3CBAAK1
SCHEMBL13026231 0.85 CYP3A4 (0.47) CYP3A4
SCHEMBL13026228 0.83 AAK1 (0.35) CTSBPPP3CBAAK1
SCHEMBL2894467 0.83 AAK1 (0.35) CTSBPPP3CBAAK1
SCHEMBL2897382 0.77 CYP3A4 (0.45) CTSBPPP3CBCYP3A4
SCHEMBL375308 0.75 CTSB (0.56) CTSBPPP3CBCYP3A4ABCC1ABCC2
SCHEMBL13668840 0.75 CTSB (0.40) CTSBPPP3CBCYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2083844-B1 HCV NS3 PROTEASE INHIBITORS MERCK SHARP & DOHME (US) 2013-11-27 EP disclosed
US-8377874-B2 HCV NS3 protease inhibitors MERCK SHARP & DOHME CORP. (US) 2013-02-19 US disclosed
US-20100286185-A1 HCV NS3 Protease Inhibitors MERCK SHARP & DOHME LLC 2010-11-11 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20100286185-A1 HCV NS3 Protease Inhibitors HAVCR2, GTF3C3, CTSC CTSB 69/4885PPP3CB 250/4885CYP3A4 154/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.