SCHEMBL28892178

SCHEMBL28892178

COc1nc2c(CBr)cccc2o1

nearest known ligand 0.39

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
ELANE P08246 3/20 0.39
CNR2 P34972 1/20 0.31
KDM4E B2RXH2 1/20 0.30
MEN1 O00255 1/20 0.30
ALDH1A1 P00352 1/20 0.30
CYP1A2 P05177 1/20 0.30
CYP2C9 P11712 1/20 0.30
HPGD P15428 1/20 0.30
CYP2C19 P33261 1/20 0.30
KMT2A Q03164 1/20 0.30
F2RL3 Q96RI0 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9768577 0.76 NQO2 (0.46) KDM4EMEN1ALDH1A1CYP1A2CYP2C9
SCHEMBL28892605 0.76 ELANE (0.49) ELANEF2RL3
SCHEMBL31213014 0.73 NQO2 (0.43) KDM4EMEN1ALDH1A1CYP1A2CYP2C9
SCHEMBL5340379 0.72 KDM4E (0.44) CNR2KDM4EALDH1A1HPGD
SCHEMBL10852711 0.71 SMN1; SMN2 (0.46) KDM4EMEN1ALDH1A1HPGDKMT2A
SCHEMBL5337672 0.70 PTPN1 (0.43) KDM4EMEN1ALDH1A1CYP2C9HPGD
SCHEMBL9756985 0.70 PLK1 (0.46) ELANEKDM4EALDH1A1CYP1A2HPGD
SCHEMBL5341017 0.70 F2RL3 (0.39) KDM4EALDH1A1HPGDF2RL3
SCHEMBL9381240 0.68 ELANE (0.34) ELANE
SCHEMBL4584082 0.68 ADA (0.47) KDM4EMEN1ALDH1A1HPGDKMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-115232144-B Nitrogen-containing condensed ring derivative, pharmaceutical composition, and preparation method and application thereof 长春金赛药业有限责任公司 2024-04-02 CN disclosed
CN-115232144-A Nitrogen-containing fused ring derivative, pharmaceutical composition, preparation method and application thereof 长春金赛药业有限责任公司 2022-10-25 CN disclosed