SCHEMBL9756985

SCHEMBL9756985

CCOC(=O)c1nc2c(CBr)cccc2o1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PLK1 P53350 1/20 0.46
CYP1A2 P05177 1/20 0.44
RAB9A P51151 3/20 0.42
MAPT P10636 3/20 0.42
NPC1 O15118 2/20 0.42
KDM4E B2RXH2 5/20 0.39
AHR P35869 1/20 0.39
HSD17B10 Q99714 3/20 0.39
ELANE P08246 1/20 0.39
ALDH1A1 P00352 3/20 0.39
CA12 O43570 1/20 0.39
CA1 P00915 1/20 0.39
CA2 P00918 1/20 0.39
CA7 P43166 1/20 0.39
CA9 Q16790 1/20 0.39
CA14 Q9ULX7 1/20 0.39
L3MBTL1 Q9Y468 1/20 0.39
GABRP O00591 1/20 0.38
GABRD O14764 1/20 0.38
GABRA1 P14867 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL18342460 0.84 CYP1A2 (0.46) PLK1CYP1A2RAB9AMAPTNPC1
SCHEMBL3616211 0.83 CYP1A2 (0.49) PLK1CYP1A2RAB9AMAPTNPC1
SCHEMBL14897914 0.81 ALDH1A1 (0.48) CYP1A2RAB9AMAPTNPC1KDM4E
SCHEMBL18342357 0.80 CYP1A2 (0.45) PLK1CYP1A2RAB9AMAPTNPC1
SCHEMBL9757082 0.79 ELANE (0.44) PLK1CYP1A2KDM4EHSD17B10ELANE
SCHEMBL28669556 0.79 CYP1A2 (0.44) PLK1CYP1A2RAB9AMAPTNPC1
SCHEMBL3621004 0.75 RAB9A (0.53) CYP1A2RAB9AMAPTNPC1KDM4E
SCHEMBL9757007 0.74 CYP4F2 (0.40) PLK1CYP1A2RAB9AMAPTNPC1
SCHEMBL9757131 0.74 MAOB (0.42) CYP1A2RAB9AMAPTNPC1KDM4E
SCHEMBL3619562 0.73 RAB9A (0.68) PLK1RAB9AMAPTNPC1KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1991019475-A2 QUINOLINYL-BENZOHETEROBICYCLIC DERIVATIVES AS ANTAGONISTS OF LEUKOTRIENE D¿4? RHONE-POULENC RORER INTERNATIONAL (HOLDINGS) INC. (US) 1991-12-26 WO disclosed