SCHEMBL28892183

SCHEMBL28892183

CCCCOc1cc(F)c(N)cc1OCc1c(OC)ccc(F)c1F

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CACNA1C Q13936 1/20 0.39
CYP1A2 P05177 1/20 0.38
CYP2C9 P11712 1/20 0.38
CYP2C19 P33261 1/20 0.38
GNRHR P30968 1/20 0.38
EGFR P00533 1/20 0.35
SMPD1 P17405 3/20 0.34
PDE4A P27815 2/20 0.34
PDE4B Q07343 2/20 0.34
PDE4C Q08493 2/20 0.34
PDE4D Q08499 2/20 0.34
GLA P06280 1/20 0.34
SMN1; SMN2 Q16637 1/20 0.34
KDM4E B2RXH2 2/20 0.34
GAA P10253 2/20 0.34
MAPT P10636 2/20 0.34
TDP1 Q9NUW8 1/20 0.34
L3MBTL1 Q9Y468 1/20 0.34
MEN1 O00255 1/20 0.34
USP2 O75604 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13577264 0.90 MAPT (0.43) CACNA1CGNRHRPDE4APDE4BPDE4C
SCHEMBL30002533 0.90 GNRHR (0.43) CACNA1CGNRHRPDE4APDE4BPDE4C
SCHEMBL4301135 0.90 GNRHR (0.43) CACNA1CGNRHRPDE4APDE4BPDE4C
SCHEMBL30002430 0.89 GNRHR (0.38) CACNA1CGNRHREGFRPDE4APDE4B
Hydrochloric Acid SCHEMBL30425693 0.89 GNRHR (0.43) CACNA1CGNRHRPDE4APDE4BPDE4C
Hydrochloric Acid SCHEMBL3100373 0.89 GNRHR (0.43) CACNA1CGNRHRPDE4APDE4BPDE4C
SCHEMBL13577269 0.85 FLT1 (0.39) CACNA1CGNRHREGFRKDM4EGAA
SCHEMBL13577279 0.85 MAPT (0.37) CACNA1CGNRHRPDE4APDE4BPDE4C
SCHEMBL13577265 0.84 CACNA1C (0.38) CACNA1CGNRHRSMN1; SMN2KDM4EGAA
SCHEMBL13577220 0.82 CACNA1C (0.40) CACNA1CGNRHRPDE4APDE4BPDE4C

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-115232144-B Nitrogen-containing condensed ring derivative, pharmaceutical composition, and preparation method and application thereof 长春金赛药业有限责任公司 2024-04-02 CN disclosed
CN-115232144-A Nitrogen-containing fused ring derivative, pharmaceutical composition, preparation method and application thereof 长春金赛药业有限责任公司 2022-10-25 CN disclosed