SCHEMBL28895015

SCHEMBL28895015

CCN1CCN(c2cc(-c3ccc(Cl)cc3)nc(-c3cccnc3)n2)CC1

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TSHR P16473 3/20 0.53
PIK3CA P42336 2/20 0.48
KIT P10721 3/20 0.48
FLT3 P36888 3/20 0.48
CYP3A4 P08684 5/20 0.48
CYP2D6 P10635 4/20 0.48
CYP2C9 P11712 3/20 0.48
CYP2C19 P33261 3/20 0.48
PIK3CB P42338 1/20 0.47
PIK3CG P48736 1/20 0.47
CYP1A2 P05177 2/20 0.46
HSD17B10 Q99714 2/20 0.46
HRH4 Q9H3N8 1/20 0.46
ALDH1A1 P00352 1/20 0.46
CLK4 Q9HAZ1 1/20 0.46
HPGD P15428 1/20 0.43
KDM4E B2RXH2 1/20 0.42
ROS1 P08922 1/20 0.42
MAPT P10636 1/20 0.42
MAPK1 P28482 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30085626 1.00 TSHR (0.53) TSHRPIK3CAKITFLT3CYP3A4
SCHEMBL28894723 0.93 CYP3A4 (0.48) TSHRPIK3CACYP3A4CYP2D6CYP2C9
SCHEMBL30085495 0.93 CYP3A4 (0.48) TSHRPIK3CACYP3A4CYP2D6CYP2C9
SCHEMBL30085522 0.88 CYP3A4 (0.61) TSHRPIK3CACYP3A4CYP2D6CYP2C9
SCHEMBL28894907 0.88 CYP3A4 (0.61) TSHRPIK3CACYP3A4CYP2D6CYP2C9
SCHEMBL30085545 0.87 CASP1 (0.50) TSHRPIK3CACYP3A4CYP2D6CYP2C9
SCHEMBL28894647 0.87 PIM1 (0.49) TSHRPIK3CACYP3A4CYP2D6CYP2C9
SCHEMBL28894632 0.87 CASP1 (0.50) TSHRPIK3CACYP3A4CYP2D6CYP2C9
SCHEMBL30085814 0.87 PIM1 (0.49) TSHRPIK3CACYP3A4CYP2D6CYP2C9
SCHEMBL28894859 0.86 HPGD (0.59) TSHRPIK3CACYP3A4CYP2D6CYP2C9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-115397818-A Aminopyrimidine derivatives and their use as modulators of arene receptors 东亚ST株式会社 2022-11-25 CN claimed
CN-115397818-A Aminopyrimidine derivatives and their use as modulators of arene receptors 东亚ST株式会社 2022-11-25 CN disclosed