SCHEMBL30085495

SCHEMBL30085495

CCCN1CCN(c2cc(-c3ccc(Cl)cc3)nc(-c3cccnc3)n2)CC1

nearest known ligand 0.51

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
CYP3A4 P08684 5/20 0.48
CYP2D6 P10635 4/20 0.48
TSHR P16473 2/20 0.48
CYP1A2 P05177 2/20 0.48
HRH4 Q9H3N8 1/20 0.48
ALDH1A1 P00352 1/20 0.48
HSD17B10 Q99714 1/20 0.48
CLK4 Q9HAZ1 1/20 0.48
PIK3CA P42336 2/20 0.47
CYP2C9 P11712 3/20 0.47
CYP2C19 P33261 3/20 0.47
PIK3CB P42338 1/20 0.47
PIK3CG P48736 1/20 0.47
ROS1 P08922 3/20 0.43
HPGD P15428 1/20 0.43
GSK3B P49841 1/20 0.42
AIMP2 Q13155 1/20 0.42
KDM4E B2RXH2 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28894723 1.00 CYP3A4 (0.48) CYP3A4CYP2D6TSHRCYP1A2HRH4
SCHEMBL30085626 0.93 TSHR (0.53) CYP3A4CYP2D6TSHRCYP1A2HRH4
SCHEMBL28895015 0.93 TSHR (0.53) CYP3A4CYP2D6TSHRCYP1A2HRH4
SCHEMBL28894647 0.91 PIM1 (0.49) CYP3A4CYP2D6TSHRCYP1A2HRH4
SCHEMBL30085814 0.91 PIM1 (0.49) CYP3A4CYP2D6TSHRCYP1A2HRH4
SCHEMBL28894784 0.90 P4HTM (0.49) CYP3A4CYP2D6TSHRCYP1A2HRH4
SCHEMBL30085370 0.90 P4HTM (0.49) CYP3A4CYP2D6TSHRCYP1A2HRH4
SCHEMBL30085539 0.90 CYP3A4 (0.60) CYP3A4CYP2D6TSHRCYP1A2HSD17B10
SCHEMBL28894649 0.90 CYP3A4 (0.60) CYP3A4CYP2D6TSHRCYP1A2HSD17B10
SCHEMBL30085522 0.89 CYP3A4 (0.61) CYP3A4CYP2D6TSHRCYP1A2HRH4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-115397818-A Aminopyrimidine derivatives and their use as modulators of arene receptors 东亚ST株式会社 2022-11-25 CN claimed
CN-115397818-A Aminopyrimidine derivatives and their use as modulators of arene receptors 东亚ST株式会社 2022-11-25 CN disclosed