SCHEMBL28895174

SCHEMBL28895174

Clc1ccc(-c2cc(NCc3ccncc3)nc(-c3cccnc3)n2)cc1

nearest known ligand 0.64

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CLK4 Q9HAZ1 8/20 0.64
DYRK1A Q13627 3/20 0.64
CYP3A4 P08684 7/20 0.56
CYP2C9 P11712 2/20 0.56
ALDH1A1 P00352 4/20 0.53
PDE5A O76074 3/20 0.53
SMN1; SMN2 Q16637 2/20 0.53
LMNA P02545 2/20 0.53
KDM4E B2RXH2 1/20 0.53
HTT P42858 1/20 0.53
NPSR1 Q6W5P4 1/20 0.53
CYP1A2 P05177 5/20 0.52
CYP2D6 P10635 5/20 0.52
CYP2C19 P33261 4/20 0.52
USP2 O75604 2/20 0.52
ALOX15 P16050 2/20 0.50
HSD17B10 Q99714 3/20 0.48
TSHR P16473 2/20 0.47
HPGD P15428 1/20 0.47
TDP1 Q9NUW8 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30085882 1.00 CLK4 (0.64) CLK4DYRK1ACYP3A4CYP2C9ALDH1A1
SCHEMBL30085785 0.92 ALDH1A1 (0.62) CLK4DYRK1ACYP3A4CYP2C9ALDH1A1
SCHEMBL28959741 0.92 ALDH1A1 (0.62) CLK4DYRK1ACYP3A4CYP2C9ALDH1A1
SCHEMBL28895256 0.84 CYP3A4 (0.57) CLK4DYRK1ACYP3A4CYP2C9ALDH1A1
SCHEMBL30085796 0.84 CYP3A4 (0.57) CLK4DYRK1ACYP3A4CYP2C9ALDH1A1
SCHEMBL28894839 0.83 CYP3A4 (0.59) CLK4DYRK1ACYP3A4CYP2C9ALDH1A1
SCHEMBL30085777 0.83 CYP3A4 (0.59) CLK4DYRK1ACYP3A4CYP2C9ALDH1A1
SCHEMBL28895149 0.82 CYP3A4 (0.55) CLK4DYRK1ACYP3A4CYP2C9ALDH1A1
SCHEMBL28894899 0.82 DYRK1A (0.53) CLK4DYRK1ACYP3A4CYP2C9ALDH1A1
SCHEMBL30085872 0.82 CYP3A4 (0.55) CLK4DYRK1ACYP3A4CYP2C9ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-115397818-A Aminopyrimidine derivatives and their use as modulators of arene receptors 东亚ST株式会社 2022-11-25 CN disclosed