SCHEMBL28896351

SCHEMBL28896351

Brc1ccc(CC(NC2CC2)c2ccccc2)cc1

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SLC18A3 Q16572 2/20 0.40
CYP1A2 P05177 1/20 0.40
CYP3A4 P08684 1/20 0.40
CYP2D6 P10635 1/20 0.40
CYP2C9 P11712 1/20 0.40
CYP2C19 P33261 1/20 0.40
L3MBTL1 Q9Y468 2/20 0.39
GAA P10253 1/20 0.39
SIGMAR1 Q99720 2/20 0.39
HTR2A P28223 1/20 0.39
NPSR1 Q6W5P4 3/20 0.38
LMNA P02545 2/20 0.38
BCHE P06276 1/20 0.38
ACHE P22303 1/20 0.38
BACE1 P56817 1/20 0.38
HTT P42858 2/20 0.38
ALDH1A1 P00352 1/20 0.38
NCOA1 Q15788 1/20 0.38
SMN1; SMN2 Q16637 1/20 0.38
NCOA3 Q9Y6Q9 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL18952114 0.94 MMP2 (0.40) SLC18A3CYP1A2CYP3A4CYP2D6CYP2C9
SCHEMBL28426623 0.84 MEN1 (0.41) CYP1A2CYP3A4CYP2D6CYP2C9CYP2C19
SCHEMBL28428823 0.84 SIGMAR1 (0.43) CYP1A2CYP3A4CYP2D6CYP2C9CYP2C19
SCHEMBL18952149 0.78 SLC6A4 (0.43) CYP1A2CYP3A4CYP2D6CYP2C9CYP2C19
SCHEMBL2021082 0.72 CYP1A2 (0.44) SLC18A3CYP1A2CYP3A4CYP2D6CYP2C9
SCHEMBL14209227 0.72 HTR2A (0.57) SIGMAR1HTR2AALDH1A1KMT2ASLC6A4
SCHEMBL28496737 0.71 KDM1A (0.44) CYP1A2CYP3A4CYP2D6CYP2C9CYP2C19
Hydrochloric Acid SCHEMBL9195769 0.70 CYP1A2 (0.50) CYP1A2CYP3A4CYP2D6L3MBTL1SIGMAR1
Hydrochloric Acid SCHEMBL8976093 0.70 CYP1A2 (0.50) CYP1A2CYP3A4CYP2D6L3MBTL1SIGMAR1
Hydrochloric Acid SCHEMBL9195452 0.70 CYP1A2 (0.50) CYP1A2CYP3A4CYP2D6L3MBTL1SIGMAR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-105283177-B Cyclopropylamine derivatives useful as inhibitors of histone demethylase KDM1A 欧洲肿瘤研究所有限责任公司 2020-07-24 CN claimed
CN-105283177-B Cyclopropylamine derivatives useful as inhibitors of histone demethylase KDM1A 欧洲肿瘤研究所有限责任公司 2020-07-24 CN disclosed