SCHEMBL28896607

SCHEMBL28896607

CCOC(=O)NC(=S)N(CCOC1(C)CCN(C(=O)OC(C)(C)C)C1)c1cc[nH]c1C(=O)OCC

nearest known ligand 0.38

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
ATM Q13315 1/20 0.38
MAPT P10636 1/20 0.35
NPSR1 Q6W5P4 1/20 0.35
ALOX15 P16050 1/20 0.34
JAK1 P23458 8/20 0.32
JAK2 O60674 3/20 0.31
JAK3 P52333 1/20 0.31
GPR119 Q8TDV5 1/20 0.31
LMNA P02545 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29211296 0.94 ATM (0.34) ATMMAPTNPSR1ALOX15JAK1
SCHEMBL28896496 0.86 ATM (0.34) ATMMAPTNPSR1ALOX15JAK1
SCHEMBL28896615 0.78 CA12 (0.31)
SCHEMBL28896565 0.78 CA12 (0.31)
SCHEMBL28896552 0.77 ATM (0.41) ATMMAPTNPSR1ALOX15JAK1
SCHEMBL28896539 0.77 CA12 (0.30)
SCHEMBL29211265 0.76 CA12 (0.30)
SCHEMBL28896225 0.76 ADORA2B (0.31) ATMNPSR1
SCHEMBL28896332 0.76 CA12 (0.35) MAPTJAK1JAK3
SCHEMBL28896186 0.74 ADORA2B (0.30)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-115403584-B 2-thio-2, 3-dihydropyrimidine-4-one derivatives, pharmaceutical compositions, preparation methods and applications thereof 长春金赛药业有限责任公司 2024-04-02 CN disclosed
CN-115403584-A 2-thio-2, 3-dihydropyrimidine-4-one derivative, pharmaceutical composition, preparation method and application thereof 长春金赛药业有限责任公司 2022-11-29 CN disclosed