SCHEMBL28898137

SCHEMBL28898137

Cc1c(C(=O)O)c(C)n(C)c1C(=O)C(=O)NC(CF)C(F)F

nearest known ligand 0.39

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
USP2 O75604 1/20 0.39
KMT2A Q03164 1/20 0.35
NPC1 O15118 1/20 0.30
MAPT P10636 1/20 0.30
RAB9A P51151 1/20 0.30
SMN1; SMN2 Q16637 1/20 0.30
HPGD P15428 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28484401 0.88
SCHEMBL28898150 0.80 TSHR (0.42) USP2KMT2ANPC1MAPTRAB9A
SCHEMBL25645225 0.79 USP2 (0.42) USP2KMT2ANPC1MAPTRAB9A
SCHEMBL28898147 0.78 TSHR (0.43) USP2NPC1MAPTRAB9ASMN1; SMN2
SCHEMBL28898160 0.77 TSHR (0.42) USP2MAPTSMN1; SMN2
SCHEMBL28898144 0.76 KMT2A (0.41) USP2KMT2ANPC1MAPTRAB9A
SCHEMBL28491214 0.76 USP2 (0.38) USP2KMT2A
SCHEMBL21427958 0.76 USP2 (0.38) USP2KMT2A
SCHEMBL28898135 0.76 TSHR (0.41) USP2MAPTSMN1; SMN2
SCHEMBL28898154 0.76 SLC10A1 (0.46) NPC1RAB9ASMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-111868026-B Capsid protein assembly inhibitor containing N-heterocyclic five-membered ring, pharmaceutical composition and application thereof 正大天晴药业集团股份有限公司 2022-11-25 CN disclosed