SCHEMBL28898745

SCHEMBL28898745

CC(C)Nc1nc(N)nc(Nc2ccccc2)n1

nearest known ligand 0.83

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KCNH3 Q9ULD8 11/20 0.83
CTSK P43235 1/20 0.66
CA1 P00915 1/20 0.55
CA2 P00918 1/20 0.55
CA9 Q16790 1/20 0.55
MAPT P10636 2/20 0.54
KMT2A Q03164 2/20 0.54
NPC1 O15118 1/20 0.54
HTT P42858 1/20 0.54
RAB9A P51151 1/20 0.54
GAA P10253 2/20 0.53
KDM4E B2RXH2 1/20 0.53
MEN1 O00255 1/20 0.53
BCL6 P41182 1/20 0.51
POLB P06746 1/20 0.51
ALDH1A1 P00352 1/20 0.50
LMNA P02545 1/20 0.50
CYP3A4 P08684 1/20 0.50
THRB P10828 1/20 0.50
ALOX15 P16050 1/20 0.50

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30568835 0.91 KCNH3 (1.00) KCNH3CTSKCA1CA2CA9
SCHEMBL2253957 0.86 GAA (0.69) KCNH3MAPTKMT2ANPC1HTT
SCHEMBL14869705 0.84 KCNH3 (0.73) KCNH3CTSKCA1CA2CA9
SCHEMBL1924308 0.83 KCNH3 (0.83) KCNH3CTSKMAPTKMT2ANPC1
SCHEMBL30568861 0.83 KCNH3 (0.83) KCNH3CTSKMAPTKMT2ANPC1
SCHEMBL14869794 0.83 KCNH3 (0.77) KCNH3CTSKMAPTKMT2ANPC1
SCHEMBL14869760 0.82 POLB (0.61) KCNH3CTSKCA1CA2CA9
SCHEMBL15102338 0.82 KCNH3 (0.81) KCNH3CTSKCA1CA2CA9
SCHEMBL19486673 0.82 KCNH3 (0.81) KCNH3CTSKCA1CA2CA9
SCHEMBL183118 0.82 NPC1 (0.68) KCNH3CA1CA2CA9MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-111662242-B Heterocyclic IDH mutant inhibitor, preparation method and application thereof 中国药科大学 2023-10-24 CN disclosed
CN-111662242-A Heterocyclic IDH mutant inhibitor, preparation method and application thereof 中国药科大学 2020-09-15 CN disclosed