SCHEMBL28899149

SCHEMBL28899149

O=C1NCCc2cc(Br)c([N+](=O)[O-])cc21

nearest known ligand 0.66

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 1/20 0.66
MAPT P10636 1/20 0.66
PARP10 Q53GL7 13/20 0.50
PARP11 Q9NR21 9/20 0.50
PARP1 P09874 6/20 0.50
KDM4E B2RXH2 1/20 0.45
TYMS P04818 1/20 0.43
F7 P08709 1/20 0.43
F3 P13726 1/20 0.43
PDPK1 O15530 1/20 0.40
GRM5 P41594 2/20 0.38
MKNK1 Q9BUB5 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27087781 0.82 KDM4E (0.45) ALDH1A1MAPTPARP10PARP11PARP1
SCHEMBL17064696 0.82 PARP10 (0.50) ALDH1A1MAPTPARP10PARP11PARP1
SCHEMBL18875036 0.82 PARP10 (0.50) ALDH1A1MAPTPARP10PARP11PARP1
SCHEMBL31510260 0.82 KDM4E (0.45) ALDH1A1MAPTPARP10PARP11PARP1
SCHEMBL27087811 0.82 PARP10 (0.50) ALDH1A1MAPTPARP10PARP11PARP1
SCHEMBL394896 0.80 MAPT (1.00) ALDH1A1MAPTTYMS
SCHEMBL26670926 0.78 PARP10 (0.43) ALDH1A1MAPTPARP10PARP11PARP1
SCHEMBL25947347 0.78 KDM4E (0.46) ALDH1A1MAPTPARP10PARP11PARP1
SCHEMBL2205282 0.78 MEN1 (0.48) ALDH1A1MAPTPARP10PARP11PARP1
SCHEMBL1090688 0.78 ALDH1A1 (0.51) ALDH1A1MAPTTYMS

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-109456308-B Heterocyclic compounds as ASK inhibitors and their use 南京圣和药业股份有限公司 2022-11-29 CN disclosed
CN-109456308-A Heterocyclic compound and its application as ASK inhibitor 南京圣和药业股份有限公司 2019-03-12 CN disclosed