SCHEMBL28899183

SCHEMBL28899183

COc1ccc(Cn2ccc3cc(Br)c(N)cc3c2=O)cc1

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPT P10636 6/20 0.49
TP53 P04637 4/20 0.49
LMNA P02545 4/20 0.49
HDAC8 Q9BY41 6/20 0.46
HDAC6 Q9UBN7 5/20 0.46
HDAC11 Q96DB2 3/20 0.46
HDAC3 O15379 4/20 0.45
HDAC1 Q13547 4/20 0.45
HDAC2 Q92769 4/20 0.45
HDAC10 Q969S8 4/20 0.45
HDAC4 P56524 2/20 0.45
HDAC7 Q8WUI4 2/20 0.45
HDAC9 Q9UKV0 2/20 0.45
HDAC5 Q9UQL6 2/20 0.45
NCOR2 Q9Y618 1/20 0.45
POLB P06746 2/20 0.43
ROCK2 O75116 1/20 0.42
ROCK1 Q13464 1/20 0.42
RXFP1 Q9HBX9 1/20 0.42
MEN1 O00255 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30095464 1.00 MAPT (0.49) MAPTTP53LMNAHDAC8HDAC6
SCHEMBL1572340 0.87 MAPT (0.51) MAPTTP53LMNAHDAC8HDAC6
SCHEMBL2332782 0.83 LMNA (0.49) MAPTTP53LMNAHDAC8HDAC6
SCHEMBL28899182 0.82 MAPT (0.46) MAPTTP53LMNAHDAC8HDAC6
SCHEMBL1571627 0.81 MAPT (0.52) MAPTTP53LMNAHDAC8HDAC6
SCHEMBL28899173 0.81 MAPT (0.45) MAPTTP53LMNAHDAC8HDAC6
SCHEMBL1412098 0.79 LMNA (0.53) MAPTTP53LMNAHDAC8HDAC6
SCHEMBL1411575 0.77 MAPT (0.51) MAPTTP53LMNAHDAC8HDAC6
SCHEMBL1411852 0.77 LMNA (0.54) MAPTTP53LMNAHDAC8HDAC6
SCHEMBL2335472 0.76 MAPT (0.40) MAPTTP53LMNAHDAC8HDAC6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-109456308-B Heterocyclic compounds as ASK inhibitors and their use 南京圣和药业股份有限公司 2022-11-29 CN disclosed
CN-109456308-A Heterocyclic compound and its application as ASK inhibitor 南京圣和药业股份有限公司 2019-03-12 CN disclosed