SCHEMBL28900166

SCHEMBL28900166

CCNC(=O)c1nc(Cl)nc2ccsc12

nearest known ligand 0.57

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
ADORA2A P29274 17/20 0.57
ADORA2B P29275 14/20 0.57
ADORA1 P30542 5/20 0.46
ADORA3 P0DMS8 2/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20784338 0.82 ADORA2A (0.74) ADORA2AADORA2BADORA1ADORA3
SCHEMBL20784296 0.80 ADORA2B (0.56) ADORA2AADORA2BADORA1ADORA3
SCHEMBL20784693 0.78 ADORA2B (0.63) ADORA2AADORA2B
SCHEMBL3661138 0.78 ADORA2A (0.43) ADORA2AADORA2BADORA1
SCHEMBL16505979 0.77 CDK9 (0.48) ADORA2AADORA2BADORA1
SCHEMBL24261174 0.77 ADORA2A (0.66) ADORA2AADORA2BADORA1ADORA3
SCHEMBL20784326 0.77 ADORA2A (0.54) ADORA2AADORA2B
SCHEMBL20784717 0.76 ADORA2A (0.78) ADORA2AADORA2BADORA1ADORA3
SCHEMBL20785049 0.76 ADORA2B (0.41) ADORA2AADORA2BADORA1ADORA3
SCHEMBL20784725 0.75 ADORA2B (0.77) ADORA2AADORA2BADORA1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-111629728-A Compounds and methods for modulating adenosine A2B receptor and adenosine A2A receptor 科尔沃斯制药股份有限公司 2020-09-04 CN disclosed