SCHEMBL28900699

SCHEMBL28900699

O=C(O)c1ccc(Br)cc1OC(CF)C(F)F

nearest known ligand 0.38

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 2/20 0.38
GLA P06280 1/20 0.38
SLC6A4 P31645 1/20 0.38
PTGER1 P34995 3/20 0.36
CFD P00746 1/20 0.36
MYC P01106 1/20 0.36
NR4A1 P22736 1/20 0.36
TDP1 Q9NUW8 1/20 0.35
PTGDR2 Q9Y5Y4 2/20 0.35
APEX1 P27695 1/20 0.35
POLB P06746 1/20 0.35
DGAT1 O75907 1/20 0.34
ALDH1A1 P00352 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28953508 1.00 KDM4E (0.38) KDM4EGLASLC6A4PTGER1CFD
SCHEMBL28953472 0.87 SLC6A4 (0.34) SLC6A4PTGDR2DGAT1
SCHEMBL28900742 0.85 GAA (0.40) KDM4ETDP1ALDH1A1
SCHEMBL5236256 0.82 KDM4E (0.44) KDM4EGLAPTGER1CFDMYC
SCHEMBL28953476 0.80 TSHR (0.38) PTGER1
SCHEMBL20107872 0.79 ALDH1A1 (0.41) KDM4EGLACFDMYCNR4A1
SCHEMBL29816552 0.79 ALDH1A1 (0.41) KDM4EGLACFDMYCNR4A1
SCHEMBL28953507 0.78 DHODH (0.42)
SCHEMBL20242123 0.75 ALDH1A1 (0.54) KDM4EGLACFDMYCNR4A1
SCHEMBL28953505 0.74 GPR17 (0.31) ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-115427109-A Heterocyclic compounds as dihydroorotate dehydrogenase inhibitors 詹森生物科技公司 2022-12-02 CN disclosed