SCHEMBL28900930

SCHEMBL28900930

COc1cc2ncnc(Oc3cc(F)c(C(=O)C(=O)Nc4ccc(Br)cc4)c(F)c3)c2cc1OC

nearest known ligand 0.69

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
KDR P35968 18/20 0.69
PDGFRA P16234 1/20 0.62
MET P08581 2/20 0.59
RAF1 P04049 1/20 0.59
PDGFRB P09619 1/20 0.59
KIT P10721 1/20 0.59
SRC P12931 1/20 0.59
FLT1 P17948 1/20 0.59
FLT4 P35916 1/20 0.59
CSF1R P07333 1/20 0.57
EGFR P00533 1/20 0.57
BRAF P15056 2/20 0.53

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30447715 0.93 KDR (0.71) KDRPDGFRAMETRAF1PDGFRB
SCHEMBL30448158 0.93 MET (0.65) KDRPDGFRAMETRAF1CSF1R
SCHEMBL28900931 0.89 KDR (0.57) KDRPDGFRAMETRAF1PDGFRB
SCHEMBL30448135 0.89 KDR (0.57) KDRPDGFRAMETRAF1PDGFRB
SCHEMBL28473758 0.88 KDR (0.59) KDRPDGFRAMETRAF1PDGFRB
SCHEMBL30447680 0.88 KDR (0.58) KDRPDGFRAMETRAF1PDGFRB
SCHEMBL28476822 0.87 KDR (0.74) KDRPDGFRARAF1PDGFRBFLT1
SCHEMBL30448047 0.87 KDR (0.74) KDRPDGFRARAF1PDGFRBFLT1
SCHEMBL28471921 0.87 KDR (0.57) KDRPDGFRAMETRAF1PDGFRB
SCHEMBL30447991 0.86 KDR (0.61) KDRPDGFRAMETRAF1PDGFRB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-111825605-B Aryl ketone amide compound and preparation method and application thereof 中国科学院上海药物研究所 2023-03-31 CN disclosed
CN-111825605-A Aryl ketone amide compound and preparation method and application thereof 中国科学院上海药物研究所 2020-10-27 CN disclosed