SCHEMBL30447680

SCHEMBL30447680

COc1cc2ncnc(Oc3cc(F)c(C(=O)C(=O)Nc4ccc([N+](=O)[O-])cc4)c(F)c3)c2cc1OC

nearest known ligand 0.58

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
KDR P35968 15/20 0.58
PDGFRA P16234 3/20 0.58
CSF1R P07333 1/20 0.54
MET P08581 2/20 0.53
ABCG2 Q9UNQ0 1/20 0.52
PDGFRB P09619 1/20 0.52
KIT P10721 1/20 0.52
FLT3 P36888 1/20 0.52
BRAF P15056 3/20 0.50
RAF1 P04049 1/20 0.49
MAPK14 Q16539 1/20 0.49
TNNI3K Q59H18 1/20 0.49

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30447813 0.91 KDR (0.56) KDRPDGFRACSF1RMETABCG2
SCHEMBL30447715 0.90 KDR (0.71) KDRPDGFRACSF1RMETPDGFRB
SCHEMBL30448158 0.89 MET (0.65) KDRPDGFRACSF1RMETBRAF
SCHEMBL28900930 0.88 KDR (0.69) KDRPDGFRACSF1RMETPDGFRB
SCHEMBL28979425 0.86 BRAF (0.56) KDRPDGFRABRAFRAF1MAPK14
SCHEMBL30447912 0.86 BRAF (0.56) KDRPDGFRABRAFRAF1MAPK14
SCHEMBL28473758 0.85 KDR (0.59) KDRPDGFRACSF1RMETPDGFRB
SCHEMBL28476822 0.84 KDR (0.74) KDRPDGFRACSF1RPDGFRBBRAF
SCHEMBL30448047 0.84 KDR (0.74) KDRPDGFRACSF1RPDGFRBBRAF
SCHEMBL28471921 0.84 KDR (0.57) KDRPDGFRACSF1RMETPDGFRB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-111825605-B Aryl ketone amide compound and preparation method and application thereof 中国科学院上海药物研究所 2023-03-31 CN disclosed