SCHEMBL28901137

SCHEMBL28901137

CC(C)(C)OC(=O)NC(=O)C=CCBr

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CTSK P43235 3/20 0.38
CA2 P00918 2/20 0.37
CA12 O43570 2/20 0.37
CA14 Q9ULX7 2/20 0.37
TDP1 Q9NUW8 1/20 0.36
CA1 P00915 2/20 0.35
CA7 P43166 2/20 0.35
MEN1 O00255 1/20 0.34
GAA P10253 1/20 0.34
KMT2A Q03164 1/20 0.34
AKT1 P31749 1/20 0.34
APLNR P35414 1/20 0.33
NPC1 O15118 1/20 0.33
RECQL P46063 1/20 0.33
RAB9A P51151 1/20 0.33
SMN1; SMN2 Q16637 1/20 0.33
NFKB1 P19838 1/20 0.33
NFKB2 Q00653 1/20 0.33
RELA Q04206 1/20 0.33
MAOA P21397 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5409226 0.79 CTSK (0.45) CTSKCA2CA12CA14TDP1
SCHEMBL5409221 0.79 CTSK (0.45) CTSKCA2CA12CA14TDP1
SCHEMBL15739550 0.77 TDP1 (0.38) CTSKCA2CA12CA14TDP1
SCHEMBL6759476 0.76 HDAC6 (0.32) CTSKCA2CA12CA14DGAT1
SCHEMBL6759479 0.76 HDAC6 (0.32) CTSKCA2CA12CA14DGAT1
SCHEMBL31430383 0.76 CTSK (0.41) CTSKCA2CA12CA14TDP1
SCHEMBL2877516 0.76 CTSK (0.39) CTSKCA2CA12CA14TDP1
SCHEMBL22288334 0.74 TDP1 (0.43) CTSKCA2CA12CA14TDP1
SCHEMBL28454875 0.74 TDP1 (0.43) CTSKCA2CA12CA14TDP1
SCHEMBL22884398 0.73 CA12 (0.30) CA2CA12CA14

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-111718361-A Metal beta-lactamase inhibitor and preparation method and application thereof 南京工业大学 2020-09-29 CN claimed
CN-111718361-B Metal beta-lactamase inhibitor and preparation method and application thereof 南京工业大学 2022-04-05 CN disclosed
CN-111718361-A Metal beta-lactamase inhibitor and preparation method and application thereof 南京工业大学 2020-09-29 CN disclosed