SCHEMBL28901544

SCHEMBL28901544

CO[Si](CCOCOc1ccc(-c2nnc(S)n2Cc2ccccc2)cc1)(OC)OC

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MEN1 O00255 2/20 0.43
KMT2A Q03164 2/20 0.43
ALDH1A1 P00352 4/20 0.42
HTT P42858 3/20 0.42
HPGD P15428 3/20 0.42
MAPT P10636 3/20 0.42
NPSR1 Q6W5P4 3/20 0.42
SMN1; SMN2 Q16637 2/20 0.42
TP53 P04637 1/20 0.42
PDE6D O43924 6/20 0.40
L3MBTL1 Q9Y468 2/20 0.40
NPC1 O15118 1/20 0.40
RAB9A P51151 1/20 0.40
KDM4E B2RXH2 3/20 0.38
LMNA P02545 2/20 0.38
CNR2 P34972 1/20 0.38
GABRA1 P14867 1/20 0.38
GABRG2 P18507 1/20 0.38
GABRB3 P28472 1/20 0.38
GABRA5 P31644 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1104386 0.83 ALDH1A1 (0.59) MEN1KMT2AALDH1A1HTTHPGD
SCHEMBL28485108 0.81 PDE6D (0.59) MEN1KMT2AALDH1A1PDE6DNPC1
SCHEMBL28489555 0.77 PDE6D (0.55) MEN1KMT2AALDH1A1HTTHPGD
SCHEMBL1104378 0.75 ALDH1A1 (0.54) MEN1KMT2AALDH1A1HTTHPGD
SCHEMBL1104400 0.74 ALDH1A1 (0.50) KMT2AALDH1A1HTTHPGDNPSR1
SCHEMBL28489558 0.73 PDE1A (0.43) MEN1KMT2AALDH1A1HTTHPGD
SCHEMBL10011720 0.72 PDE4A (0.49) MEN1KMT2AALDH1A1HPGDMAPT
SCHEMBL1104402 0.72 ALDH1A1 (0.55) KMT2AALDH1A1HPGDMAPTNPSR1
SCHEMBL10480335 0.71 ALDH1A1 (0.55) MEN1KMT2AALDH1A1HPGDMAPT
SCHEMBL1104406 0.71 MEN1 (0.55) MEN1KMT2AALDH1A1HTTHPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-111875583-B Triazole derivative and preparation method and application thereof 中国科学院上海药物研究所 2021-06-15 CN disclosed
CN-109666022-B Triazole derivative and preparation method and application thereof 中国科学院上海药物研究所 2021-06-15 CN disclosed
CN-111875583-A Triazole derivative and preparation method and application thereof 中国科学院上海药物研究所 2020-11-03 CN disclosed