SCHEMBL28905313

SCHEMBL28905313

CC(C)(C)NC(=O)O[C@@H]1c2cc(F)ccc2CC12CCNCC2

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
DPP4 P27487 1/20 0.38
ACHE P22303 3/20 0.35
BCHE P06276 1/20 0.34
CCNE1 P24864 1/20 0.33
CDK2 P24941 1/20 0.33
HTR2A P28223 1/20 0.33
HTR2C P28335 1/20 0.33
CCNT1 O60563 1/20 0.33
CDK9 P50750 1/20 0.33
KDM1A O60341 2/20 0.32
SLC9A3 P48764 1/20 0.32
CYP2D6 P10635 3/20 0.31
SLC6A2 P23975 2/20 0.31
SLC6A4 P31645 2/20 0.31
SLC6A3 Q01959 1/20 0.31
SSTR4 P31391 1/20 0.31
DPP8 Q6V1X1 2/20 0.31
DPP9 Q86TI2 2/20 0.31
CHRM2 P08172 2/20 0.31
CHRM1 P11229 2/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28513992 0.92 DPP4 (0.38) DPP4ACHEBCHECCNE1CDK2
SCHEMBL28511456 0.84 DPP9 (0.34) ACHEBCHECYP2D6SLC6A2SLC6A4
SCHEMBL29891133 0.77 RORC (0.37) DPP4HTR2AHTR2CKDM1ADPP8
SCHEMBL23046128 0.77 RORC (0.37) DPP4HTR2AHTR2CKDM1ADPP8
SCHEMBL21397469 0.75 DPP4 (0.37) DPP4HTR2AHTR2CSLC9A3SLC6A2
SCHEMBL21383892 0.71 DPP4 (0.40) DPP4HTR2AHTR2CKDM1ACYP2D6
SCHEMBL29891089 0.70 NPY5R (0.36) DPP4KDM1ACYP2D6DPP8DPP9
SCHEMBL23046130 0.70 NPY5R (0.36) DPP4KDM1ACYP2D6DPP8DPP9
SCHEMBL21383810 0.69 HTR2C (0.41) DPP4HTR2AHTR2CKDM1ASLC6A2
SCHEMBL29726234 0.69 HTR2C (0.41) DPP4HTR2AHTR2CKDM1ASLC6A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-117263942-A SHP2 phosphatase inhibitors and methods of use thereof 传达治疗有限公司 2023-12-22 CN disclosed
CN-112166110-B SHP2 phosphatase inhibitors and methods of use thereof 传达治疗有限公司 2023-08-11 CN disclosed
CN-112166110-A SHP2 phosphatase inhibitors and methods of use thereof 传达治疗有限公司 2021-01-01 CN disclosed