SCHEMBL21397469

SCHEMBL21397469

CC(C)(C)OC(=O)[C@@H]1c2cc(F)ccc2CC12CCNCC2

nearest known ligand 0.37

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
DPP4 P27487 1/20 0.37
HTR2A P28223 1/20 0.35
HTR2C P28335 1/20 0.35
DPP8 Q6V1X1 3/20 0.34
DPP9 Q86TI2 2/20 0.34
NR3C2 P08235 1/20 0.33
SLC9A3 P48764 1/20 0.33
SLC6A4 P31645 4/20 0.32
SLC6A2 P23975 3/20 0.32
GABRA1 P14867 1/20 0.31
GABRG2 P18507 1/20 0.31
GABRB3 P28472 1/20 0.31
GABRA5 P31644 1/20 0.31
GABRA3 P34903 1/20 0.31
GABRA2 P47869 1/20 0.31
GABRA4 P48169 1/20 0.31
GABRA6 Q16445 1/20 0.31
NR1H2 P55055 1/20 0.30
BRD3 Q15059 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21397429 0.91 DPP4 (0.37) DPP4HTR2AHTR2CDPP8DPP9
SCHEMBL23046128 0.81 RORC (0.37) DPP4HTR2AHTR2CDPP8DPP9
SCHEMBL29891133 0.81 RORC (0.37) DPP4HTR2AHTR2CDPP8DPP9
SCHEMBL23046130 0.75 NPY5R (0.36) DPP4DPP8DPP9NR3C2
SCHEMBL28905313 0.75 DPP4 (0.38) DPP4HTR2AHTR2CDPP8DPP9
SCHEMBL29891089 0.75 NPY5R (0.36) DPP4DPP8DPP9NR3C2
SCHEMBL21383892 0.71 DPP4 (0.40) DPP4HTR2AHTR2C
SCHEMBL21383810 0.71 HTR2C (0.41) DPP4HTR2AHTR2CSLC6A4SLC6A2
SCHEMBL29726234 0.71 HTR2C (0.41) DPP4HTR2AHTR2CSLC6A4SLC6A2
SCHEMBL25991491 0.71 HTR2C (0.41) DPP4HTR2AHTR2CSLC6A4SLC6A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2019183367-A1 SHP2 PHOSPHATASE INHIBITORS AND METHODS OF USE THEREOF RELAY THERAPEUTICS, INC. (US) 2019-09-26 WO disclosed