SCHEMBL28906373

SCHEMBL28906373

c1csc(-c2[nH]c3ccccc3c2Cc2c(-c3cccs3)[nH]c3ccccc23)c1

nearest known ligand 0.62

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
DRD2 P14416 1/20 0.62
HTR2A P28223 1/20 0.62
HTR2C P28335 1/20 0.62
KDM4E B2RXH2 4/20 0.54
GAA P10253 2/20 0.49
CNR1 P21554 1/20 0.48
ALDH1A1 P00352 5/20 0.47
MAPT P10636 4/20 0.47
MEN1 O00255 3/20 0.47
KMT2A Q03164 3/20 0.47
LMNA P02545 3/20 0.47
PPARG P37231 2/20 0.47
NCOA2 Q15596 2/20 0.47
NCOA1 Q15788 2/20 0.47
NPSR1 Q6W5P4 1/20 0.47
NCOA3 Q9Y6Q9 1/20 0.47
TDO2 P48775 1/20 0.47
KCNH2 Q12809 1/20 0.46
HDAC1 Q13547 1/20 0.46
TUBB4A P04350 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9272303 0.81 HTR2A (0.57) DRD2HTR2AHTR2CKDM4EGAA
SCHEMBL6281078 0.79 KDM4E (0.56) DRD2HTR2AHTR2CKDM4EGAA
SCHEMBL27543191 0.77 DRD2 (0.52) DRD2HTR2AHTR2CKDM4EGAA
SCHEMBL29955809 0.77 KDM4E (0.51) DRD2HTR2AHTR2CKDM4EGAA
SCHEMBL29218370 0.76 KDM4E (0.50) DRD2HTR2AHTR2CKDM4EGAA
SCHEMBL28253382 0.75 ESR1 (0.62) DRD2HTR2AHTR2CKDM4ECNR1
SCHEMBL5419527 0.73 DRD2 (0.51) DRD2HTR2AHTR2CKDM4EALDH1A1
SCHEMBL28906516 0.72 HTR2A (0.62) DRD2HTR2AHTR2CCNR1TUBB4A
SCHEMBL28254266 0.71 ESR1 (0.49) DRD2HTR2AHTR2CKDM4EGAA
SCHEMBL7039033 0.70 ESR1 (0.67) DRD2HTR2AHTR2CKDM4EGAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-115304533-B Bisindolemethane type alpha-glucosidase inhibitor and preparation method and application thereof 中国医学科学院药用植物研究所云南分所 2024-04-12 CN disclosed
CN-117567447-A Thiophene-containing bis-indolomethane type a-glucosidase inhibitor and preparation method and application thereof 中国医学科学院药用植物研究所云南分所 2024-02-20 CN disclosed
CN-115304533-A Bis-indole methane type alpha-glucosidase inhibitor and preparation method and application thereof 中国医学科学院药用植物研究所云南分所 2022-11-08 CN disclosed