SCHEMBL28907820

SCHEMBL28907820

CC(C)(C)OC(=O)n1ccc(-c2ccc3c(c2)NC(=O)CO3)c1

nearest known ligand 0.45

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 4/20 0.45
ALDH1A1 P00352 4/20 0.45
RAB9A P51151 3/20 0.45
NPC1 O15118 2/20 0.45
SMN1; SMN2 Q16637 1/20 0.45
PDE3B Q13370 1/20 0.44
PDE3A Q14432 1/20 0.44
MMP12 P39900 1/20 0.44
NR3C2 P08235 5/20 0.44
MAPT P10636 3/20 0.43
TRPV1 Q8NER1 4/20 0.42
PARP1 P09874 1/20 0.42
NR3C1 P04150 1/20 0.41
PGR P06401 1/20 0.41
HPGD P15428 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL18305033 0.83 NR3C2 (0.49) KDM4EALDH1A1RAB9ANPC1SMN1; SMN2
SCHEMBL28909618 0.82 NR3C2 (0.43) NR3C2TRPV1NR3C1PGR
SCHEMBL12405056 0.80 NR3C2 (0.48) KDM4EALDH1A1RAB9ANPC1SMN1; SMN2
SCHEMBL23830447 0.72 TRPV1 (0.45) ALDH1A1SMN1; SMN2MMP12NR3C2MAPT
SCHEMBL13343865 0.71 BRD4 (0.57) KDM4EALDH1A1MAPTPARP1HPGD
SCHEMBL5362061 0.71 DRD4 (0.59) PARP1
SCHEMBL29120487 0.71 ALDH1A1 (0.59) ALDH1A1MMP12MAPTTRPV1
SCHEMBL30674772 0.71 ALDH1A1 (0.59) ALDH1A1MMP12MAPTTRPV1
SCHEMBL28907822 0.70 PDE4B (0.52) KDM4EALDH1A1SMN1; SMN2MMP12NR3C2
SCHEMBL4180037 0.70 HRH3 (0.54) TRPV1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-107873031-B Benzoxazinone derivatives and analogs thereof as modulators of TNF activity UCB生物制药私人有限公司 2021-03-12 CN disclosed