SCHEMBL28909618

SCHEMBL28909618

CC(C)(C)OC(=O)n1ccc(-c2cc(F)c3c(c2)NC(=O)CO3)c1

nearest known ligand 0.43

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
NR3C2 P08235 8/20 0.43
PGR P06401 7/20 0.43
NR3C1 P04150 6/20 0.43
AR P10275 1/20 0.34
HTR1A P08908 3/20 0.34
HTR1D P28221 1/20 0.34
HTR1B P28222 1/20 0.34
SLC6A4 P31645 1/20 0.34
BRD4 O60885 3/20 0.33
CREBBP Q92793 3/20 0.33
ADRB2 P07550 3/20 0.33
DRD2 P14416 2/20 0.33
HTR2A P28223 2/20 0.33
ADRB1 P08588 1/20 0.33
CRBN Q96SW2 1/20 0.33
LIPC P11150 1/20 0.32
LIPG Q9Y5X9 1/20 0.32
TRPV1 Q8NER1 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL18305166 0.84 NR3C2 (0.45) NR3C2PGRNR3C1ARHTR1A
SCHEMBL28907820 0.82 KDM4E (0.45) NR3C2PGRNR3C1TRPV1
SCHEMBL28533641 0.81 CREBBP (0.35) BRD4CREBBPDRD2LIPCLIPG
SCHEMBL13343850 0.72 BRD4 (0.54) NR3C2PGRNR3C1HTR1ABRD4
SCHEMBL28525830 0.71 KDM4E (0.43) CRBN
SCHEMBL4265400 0.70 NR3C2 (0.53) NR3C2PGRNR3C1HTR1AHTR1D
SCHEMBL8195296 0.69 BRD4 (0.43) NR3C2PGRNR3C1HTR1AHTR1D
SCHEMBL4262107 0.68 NR3C2 (0.51) NR3C2PGRNR3C1HTR1AHTR1D
SCHEMBL14079839 0.66 ADRB2 (0.39) NR3C2PGRNR3C1HTR1AHTR1D
SCHEMBL4289205 0.66 NR3C2 (0.45) NR3C2PGRNR3C1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-107873031-B Benzoxazinone derivatives and analogs thereof as modulators of TNF activity UCB生物制药私人有限公司 2021-03-12 CN disclosed