SCHEMBL28909421

SCHEMBL28909421

CCn1c(=O)sc2cc(Br)ccc21

nearest known ligand 0.54

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
SIGMAR1 Q99720 7/20 0.54
MAPT P10636 3/20 0.45
SMN1; SMN2 Q16637 1/20 0.45
TP53 P04637 1/20 0.44
ADRA2A P08913 1/20 0.42
ADRA2B P18089 1/20 0.42
ADRA2C P18825 1/20 0.42
HRH1 P35367 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14681114 0.87 SIGMAR1 (0.59) SIGMAR1MAPTTP53ADRA2AADRA2B
SCHEMBL7712083 0.84 SIGMAR1 (0.63) SIGMAR1
SCHEMBL3043755 0.83 SIGMAR1 (0.54) SIGMAR1MAPTADRA2AADRA2BADRA2C
SCHEMBL17288108 0.83 SIGMAR1 (0.51) SIGMAR1MAPTSMN1; SMN2TP53ADRA2A
SCHEMBL7716707 0.83 SIGMAR1 (0.51) SIGMAR1ADRA2AADRA2BADRA2CHRH1
SCHEMBL2403333 0.81 SIGMAR1 (0.50) SIGMAR1MAPTSMN1; SMN2
SCHEMBL2073651 0.81 SIGMAR1 (0.59) SIGMAR1MAPTADRA2AADRA2BADRA2C
SCHEMBL3045443 0.80 MAPT (0.54) SIGMAR1MAPTSMN1; SMN2TP53ADRA2A
SCHEMBL11038312 0.80 MAPT (0.48) SIGMAR1MAPTSMN1; SMN2TP53ADRA2A
SCHEMBL7713334 0.78 SIGMAR1 (0.53) SIGMAR1MAPTSMN1; SMN2ADRA2AADRA2B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-113087683-B Nitrogen-substituted benzothiazolinone XOR/URAT1 dual inhibitor and preparation method and application thereof 华南理工大学 2022-04-22 CN disclosed
CN-113087683-A Nitrogen-substituted benzothiazolinone XOR/URAT1 dual inhibitor and preparation method and application thereof 华南理工大学 2021-07-09 CN disclosed