SCHEMBL28922901

SCHEMBL28922901

N#CCc1ccc2c(c1)C1(CCCCC1)CCO2

nearest known ligand 0.38

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
PIK3CA P42336 1/20 0.33
PIK3CG P48736 1/20 0.33
PDCD1 Q15116 1/20 0.33
CD274 Q9NZQ7 1/20 0.33
LMNA P02545 1/20 0.31
AKR1B1 P15121 1/20 0.31
NAAA Q02083 1/20 0.30
CYP26A1 O43174 1/20 0.30
CYP26B1 Q9NR63 1/20 0.30
KIF11 P52732 1/20 0.30
PRSS1 P07477 1/20 0.30
PRSS2 P07478 1/20 0.30
MAOA P21397 1/20 0.30
MAOB P27338 1/20 0.30
PRSS3 P35030 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30148869 0.81 LMNA (0.33) LMNAAKR1B1CYP26A1CYP26B1
SCHEMBL28922878 0.81 PDCD1 (0.36) PDCD1CD274LMNAAKR1B1CYP26A1
SCHEMBL30148890 0.77 CYP26A1 (0.48) LMNAAKR1B1CYP26A1CYP26B1
SCHEMBL28922824 0.73 KDM4E (0.40) AKR1B1
SCHEMBL30148887 0.73 KDM4E (0.40) AKR1B1
SCHEMBL1464785 0.72 CD274 (0.50) PIK3CAPIK3CGPDCD1CD274LMNA
SCHEMBL28922776 0.70 ALDH1A1 (0.44) AKR1B1
SCHEMBL4133761 0.69 CTNNB1 (0.43) PDCD1CD274MAOAMAOB
SCHEMBL4133763 0.69 KCNH2 (0.46)
SCHEMBL29790987 0.69 KCNH2 (0.46)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-115521325-A Boronic acid derivatives 首药控股(北京)股份有限公司 2022-12-27 CN disclosed