SCHEMBL28929348

SCHEMBL28929348

CCOC(=O)c1nc(-c2ccc(O)cc2)c(C)s1

nearest known ligand 0.54

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
RARA P10276 2/20 0.54
RARB P10826 2/20 0.54
RARG P13631 2/20 0.54
PTGS2 P35354 1/20 0.51
ESR1 P03372 2/20 0.49
ESR2 Q92731 2/20 0.49
CA12 O43570 1/20 0.49
CA1 P00915 1/20 0.49
CA2 P00918 1/20 0.49
CA7 P43166 1/20 0.49
CA9 Q16790 1/20 0.49
CA14 Q9ULX7 1/20 0.49
ALDH1A1 P00352 4/20 0.47
HSD17B10 Q99714 2/20 0.47
CYP1A2 P05177 2/20 0.47
CYP2C9 P11712 1/20 0.47
CYP2C19 P33261 1/20 0.47
TRPM8 Q7Z2W7 4/20 0.46
JAK2 O60674 1/20 0.45
JAK3 P52333 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28928756 0.80 ERN1 (0.44) RARARARBRARGPTGS2ALDH1A1
SCHEMBL5029389 0.76 MEN1 (0.55) RARARARBRARGPTGS2ALDH1A1
SCHEMBL5519672 0.75 PTGS2 (0.64) PTGS2ALDH1A1HSD17B10CYP1A2CYP2C9
SCHEMBL5909547 0.75 PTGS2 (0.64) PTGS2ALDH1A1HSD17B10CYP1A2CYP2C9
SCHEMBL15149783 0.75 TRPM8 (0.44) ALDH1A1CYP1A2CYP2C9CYP2C19TRPM8
SCHEMBL27356584 0.75 JAK2 (0.56) RARARARBRARGPTGS2ALDH1A1
SCHEMBL31476860 0.75 JAK2 (0.56) RARARARBRARGPTGS2ALDH1A1
SCHEMBL28928759 0.74 ESR1 (0.49) ESR1ESR2CA12CA1CA2
SCHEMBL7907788 0.74 TRPM8 (0.56) RARARARBRARGESR1ESR2
SCHEMBL5909558 0.74 PTGS2 (0.59) PTGS2ALDH1A1HSD17B10TRPM8POLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-109810073-B 4-arylthiazole derivatives and pharmaceutical compositions thereof 南京海辰药业股份有限公司 2023-01-06 CN disclosed