SCHEMBL28933993

SCHEMBL28933993

COc1ccc(C(NC(=O)C(c2ccccc2)(c2ccccc2)c2ccccc2)C(=O)O)cc1

nearest known ligand 0.54

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
ATM Q13315 1/20 0.54
NPSR1 Q6W5P4 2/20 0.48
CNR2 P34972 1/20 0.47
KCNN4 O15554 1/20 0.45
KIF11 P52732 3/20 0.44
KMT2A Q03164 2/20 0.44
ALDH1A1 P00352 2/20 0.44
TP53 P04637 1/20 0.44
CYP3A4 P08684 1/20 0.44
ACP3 P15309 1/20 0.43
MEN1 O00255 1/20 0.43
GAA P10253 1/20 0.43
GPR88 Q9GZN0 1/20 0.43
L3MBTL1 Q9Y468 1/20 0.43
TACR3 P29371 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28709110 0.89 ANPEP (0.46) ATMNPSR1CNR2KCNN4KMT2A
SCHEMBL28710172 0.89 ANPEP (0.46) ATMNPSR1CNR2KCNN4KMT2A
SCHEMBL7036247 0.82 NPSR1 (0.69) ATMNPSR1CNR2KMT2AALDH1A1
SCHEMBL28934073 0.77 HDAC3 (0.51) ATMNPSR1CNR2KMT2AALDH1A1
SCHEMBL28934074 0.77 HDAC3 (0.51) ATMNPSR1CNR2KMT2AALDH1A1
SCHEMBL11697241 0.77 ATM (0.56) ATMNPSR1CNR2KMT2AALDH1A1
SCHEMBL11646318 0.76 ATM (0.55) ATMNPSR1CNR2KMT2AALDH1A1
SCHEMBL2485730 0.75 ALDH1A1 (0.57) ATMNPSR1CNR2KMT2AALDH1A1
SCHEMBL9298424 0.75 ALDH1A1 (0.57) ATMNPSR1CNR2KMT2AALDH1A1
SCHEMBL844431 0.74 ATM (0.56) ATMNPSR1CNR2KMT2AALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-114181116-A D-amino acid derivative aminopeptidase N inhibitor and preparation method and application thereof 山东中医药大学 2022-03-15 CN disclosed