SCHEMBL28934485

SCHEMBL28934485

CS(=O)(=O)N1CCC[C@@H](Nc2nnc(-c3ccc(C#N)cc3O)c3c2CCCC3)C1

nearest known ligand 0.62

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
NLRP3 Q96P20 10/20 0.62
JAK2 O60674 8/20 0.43
JAK3 P52333 8/20 0.43
IL1B P01584 1/20 0.40
IRAK4 Q9NWZ3 1/20 0.39
JAK1 P23458 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30108806 1.00 NLRP3 (0.62) NLRP3JAK2JAK3IL1BIRAK4
SCHEMBL30108657 1.00 NLRP3 (0.62) NLRP3JAK2JAK3IL1BIRAK4
SCHEMBL28934490 1.00 NLRP3 (0.62) NLRP3JAK2JAK3IL1BIRAK4
SCHEMBL25864237 0.91 NLRP3 (0.51) NLRP3JAK2JAK3IL1BJAK1
SCHEMBL30108739 0.87 NLRP3 (0.67) NLRP3IL1B
SCHEMBL28934456 0.87 NLRP3 (0.67) NLRP3IL1B
SCHEMBL28934462 0.87 NLRP3 (0.67) NLRP3IL1B
SCHEMBL28934535 0.86 NLRP3 (0.51) NLRP3JAK2JAK3IL1BIRAK4
SCHEMBL30108776 0.86 NLRP3 (0.51) NLRP3JAK2JAK3IL1BIRAK4
SCHEMBL28934539 0.86 NLRP3 (0.51) NLRP3JAK2JAK3IL1BIRAK4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-115433163-A NLRP3 inflammasome inhibitor and application thereof 药捷安康(南京)科技股份有限公司 2022-12-06 CN disclosed