SCHEMBL28934535

SCHEMBL28934535

CS(=O)(=O)N1CCC[C@@H](Nc2nnc(-c3ccc(C#N)cc3O)c3ccccc23)C1

nearest known ligand 0.51

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
NLRP3 Q96P20 9/20 0.51
JAK2 O60674 7/20 0.43
JAK3 P52333 7/20 0.43
ALDH1A1 P00352 1/20 0.41
IRAK4 Q9NWZ3 1/20 0.41
IL1B P01584 1/20 0.40
JAK1 P23458 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30108776 1.00 NLRP3 (0.51) NLRP3JAK2JAK3ALDH1A1IRAK4
SCHEMBL28934539 1.00 NLRP3 (0.51) NLRP3JAK2JAK3ALDH1A1IRAK4
SCHEMBL28934545 0.91 NLRP3 (0.49) NLRP3JAK2ALDH1A1IRAK4IL1B
SCHEMBL25864158 0.91 NLRP3 (0.47) NLRP3JAK2JAK3ALDH1A1IL1B
SCHEMBL28934549 0.91 NLRP3 (0.49) NLRP3JAK2ALDH1A1IRAK4IL1B
SCHEMBL30108648 0.87 NLRP3 (0.62) NLRP3IL1B
SCHEMBL28934477 0.87 NLRP3 (0.62) NLRP3IL1B
SCHEMBL28934482 0.87 NLRP3 (0.62) NLRP3IL1B
SCHEMBL30108657 0.86 NLRP3 (0.62) NLRP3JAK2JAK3IRAK4IL1B
SCHEMBL30108806 0.86 NLRP3 (0.62) NLRP3JAK2JAK3IRAK4IL1B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-115433163-A NLRP3 inflammasome inhibitor and application thereof 药捷安康(南京)科技股份有限公司 2022-12-06 CN disclosed