SCHEMBL28934722

SCHEMBL28934722

CCOC(=O)c1cn(C2CCCC2)cn1

nearest known ligand 0.45

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
NOTUM Q6P988 1/20 0.45
ALDH1A1 P00352 7/20 0.43
CDK5 Q00535 3/20 0.43
CDK5R1 Q15078 3/20 0.43
TSHR P16473 1/20 0.43
SMN1; SMN2 Q16637 1/20 0.41
MAPK1 P28482 1/20 0.41
CYP1A2 P05177 1/20 0.41
POLB P06746 1/20 0.40
KDM4E B2RXH2 1/20 0.40
HPGD P15428 1/20 0.40
KDM5A P29375 1/20 0.40
CPB2 Q96IY4 2/20 0.39
KMT2A Q03164 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL22920208 0.99 ALDH1A1 (0.45) NOTUMALDH1A1CDK5CDK5R1TSHR
SCHEMBL15236764 0.99 ALDH1A1 (0.45) NOTUMALDH1A1CDK5CDK5R1TSHR
SCHEMBL12983979 0.97 NOTUM (0.45) NOTUMALDH1A1CDK5CDK5R1TSHR
SCHEMBL1268993 0.94 NOTUM (0.47) NOTUMALDH1A1CDK5CDK5R1TSHR
SCHEMBL14631229 0.89 CPB2 (0.46) NOTUMALDH1A1CDK5CDK5R1CYP1A2
SCHEMBL14631042 0.89 CPB2 (0.46) NOTUMALDH1A1CDK5CDK5R1CYP1A2
SCHEMBL14631044 0.89 CPB2 (0.46) NOTUMALDH1A1CDK5CDK5R1CYP1A2
SCHEMBL14704031 0.88 NOTUM (0.43) NOTUMALDH1A1CYP1A2KDM4EHPGD
SCHEMBL12333458 0.85 CPB2 (0.47) NOTUMALDH1A1CDK5CDK5R1CYP1A2
SCHEMBL14631486 0.85 CPB2 (0.49) NOTUMALDH1A1CDK5CDK5R1TSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-115461338-B 3-azabicyclo (3.1.0) hexane derivatives having KDM5 inhibitory activity and uses thereof 小野药品工业株式会社 2024-02-20 CN disclosed
CN-115461338-A 3-azabicyclo (3.1.0) hexane derivatives having KDM5 inhibitory activity and uses thereof 小野药品工业株式会社 2022-12-09 CN disclosed