SCHEMBL28935985

SCHEMBL28935985

CC(OC(N)=O)c1nc(-c2cccc(S(C)(=O)=O)c2)no1

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CA9 Q16790 5/20 0.44
CA2 P00918 5/20 0.44
CA12 O43570 3/20 0.44
CA1 P00915 3/20 0.44
DPP4 P27487 7/20 0.43
DPP7 Q9UHL4 7/20 0.43
FFAR1 O14842 1/20 0.41
S1PR1 P21453 1/20 0.40
TSHR P16473 1/20 0.40
MAPK1 P28482 1/20 0.40
L3MBTL1 Q9Y468 1/20 0.40
GPR119 Q8TDV5 1/20 0.40
NTRK1 P04629 1/20 0.39
MET P08581 1/20 0.39
PIM1 P11309 1/20 0.39
FGFR1 P11362 1/20 0.39
MAP2K2 P36507 1/20 0.39
FLT3 P36888 1/20 0.39
MAPK8 P45983 1/20 0.39
GSK3B P49841 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28713701 0.91 CA2 (0.55) CA9CA2CA12CA1DPP4
SCHEMBL28710978 0.84 MLLT1 (0.44) DPP4DPP7FFAR1TSHRMAPK1
SCHEMBL28706194 0.84 KCNT1 (0.49) TSHRMAPK1L3MBTL1KCNT1
SCHEMBL28710586 0.84 KCNT1 (0.49) TSHRMAPK1L3MBTL1KCNT1
SCHEMBL28706195 0.84 KCNT1 (0.49) TSHRMAPK1L3MBTL1KCNT1
SCHEMBL28710950 0.83 NPC1 (0.46) DPP4DPP7FFAR1TSHRMAPK1
SCHEMBL22637707 0.82 CA9 (0.50) CA9CA2CA12CA1DPP4
SCHEMBL22649534 0.82 CA9 (0.49) CA9CA2CA12CA1DPP4
SCHEMBL28713211 0.82 S1PR3 (0.52) CA9CA2CA12CA1FFAR1
SCHEMBL28713210 0.82 S1PR3 (0.52) CA9CA2CA12CA1FFAR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-114269340-A KCNT1 inhibitors and methods of use 普拉克西斯精密药物股份有限公司 2022-04-01 CN disclosed