SCHEMBL28945293

SCHEMBL28945293

CC(=O)Oc1ccn2ccncc12

nearest known ligand 0.36

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
BRD4 O60885 1/20 0.36
KDM4E B2RXH2 6/20 0.34
ALDH1A1 P00352 3/20 0.34
TSHR P16473 2/20 0.34
TDP1 Q9NUW8 2/20 0.34
ESR1 P03372 1/20 0.34
ITGB3 P05106 1/20 0.34
ITGA2B P08514 1/20 0.34
HMGB1 P09429 1/20 0.34
HPGD P15428 1/20 0.34
GGT1 P19440 1/20 0.34
PTGS1 P23219 1/20 0.34
PTGS2 P35354 1/20 0.34
BLM P54132 1/20 0.34
NAPRT Q6XQN6 1/20 0.34
HSD17B10 Q99714 1/20 0.34
GAA P10253 2/20 0.34
MAPT P10636 2/20 0.34
KMT2A Q03164 1/20 0.34
RAB9A P51151 3/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL28792273 0.98 BRD4 (0.36) BRD4KDM4EALDH1A1TSHRTDP1
SCHEMBL8829299 0.75 CYP3A4 (0.37) KDM4EALDH1A1TSHRTDP1GAA
SCHEMBL1424718 0.75 PTGS2 (0.44) KDM4EALDH1A1TSHRTDP1ESR1
SCHEMBL16468077 0.71 KDM4E (0.49) KDM4EALDH1A1HSD17B10GAAMAPT
SCHEMBL8829243 0.69 KDM4C (0.43) KDM4EALDH1A1TDP1NAPRTGAA
SCHEMBL3796726 0.68 SIRT3 (0.44) KDM4EALDH1A1TSHRTDP1MAPT
SCHEMBL28826867 0.68 KDM4E (0.42) BRD4KDM4EALDH1A1TSHRTDP1
SCHEMBL24656778 0.67 KDM5A (0.36) KDM4EALDH1A1GAAMAPTKMT2A
SCHEMBL10953461 0.67 TDP1 (0.47) KDM4EALDH1A1TSHRTDP1ESR1
SCHEMBL20073402 0.66 RAB9A (0.40) KDM4EALDH1A1TSHRTDP1ESR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-104144930-A New indolizine derivatives, method for preparing same and pharmaceutical compositions containing same SERVIER LAB 2014-11-12 CN disclosed
CN-102149714-A Novel tricyclic derivatives, process for the preparation thereof and pharmaceutical compositions containing same SERVIER LAB 2011-08-10 CN disclosed