SCHEMBL28947686

SCHEMBL28947686

O=S(=O)(O)C1CCC(F)(F)CC1.[NaH].[NaH]

nearest known ligand 0.44

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
TSHR P16473 2/20 0.44
LMNA P02545 1/20 0.44
CYP3A4 P08684 1/20 0.44
GABRA1 P14867 1/20 0.44
GABRG2 P18507 1/20 0.44
NFKB1 P19838 1/20 0.44
GABRB3 P28472 1/20 0.44
GABRA5 P31644 1/20 0.44
GABRA3 P34903 1/20 0.44
GABRA2 P47869 1/20 0.44
GABRA6 Q16445 1/20 0.44
EPHX2 P34913 1/20 0.33
TDP1 Q9NUW8 1/20 0.32
AKT1 P31749 1/20 0.32
PIK3CA P42336 1/20 0.32
MTOR P42345 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28947688 1.00 TSHR (0.44) TSHRLMNACYP3A4GABRA1GABRG2
SCHEMBL4318930 0.98 TSHR (0.46) TSHRLMNACYP3A4GABRA1GABRG2
SCHEMBL12520312 0.84 TSHR (0.38) TSHRLMNACYP3A4GABRA1GABRG2
SCHEMBL17159759 0.76
SCHEMBL16499932 0.75 EPHX2 (0.32) EPHX2
SCHEMBL1093575 0.73
SCHEMBL5048142 0.73 LMNA (0.46) TSHRLMNACYP3A4GABRA1GABRG2
SCHEMBL5212 0.73
SCHEMBL4620125 0.73 TSHR (0.63) TSHRLMNACYP3A4GABRA1GABRG2
SCHEMBL9991970 0.72 TSHR (0.39) TSHRLMNACYP3A4GABRA1GABRG2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-115698009-A CD73 inhibiting 2,4-dioxopyrimidine compounds 吉利德科学公司 2023-02-03 CN disclosed