SCHEMBL28947711

SCHEMBL28947711

FC(F)(F)c1cc2cc(Br)ccc2cn1

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
THRB P10828 1/20 0.44
NT5E P21589 1/20 0.44
GSK3A P49840 1/20 0.42
CDK9 P50750 1/20 0.42
CDK5 Q00535 1/20 0.42
TAOK1 Q7L7X3 1/20 0.42
CLK4 Q9HAZ1 1/20 0.42
KDM4E B2RXH2 2/20 0.39
TRPV4 Q9HBA0 1/20 0.38
CYP2A6 P11509 1/20 0.38
MEN1 O00255 1/20 0.35
ALDH1A1 P00352 1/20 0.35
MAPT P10636 1/20 0.35
KMT2A Q03164 1/20 0.35
NOS1 P29475 2/20 0.35
METAP2 P50579 2/20 0.35
BACE1 P56817 2/20 0.35
CYP1A2 P05177 1/20 0.35
CYP2C19 P33261 1/20 0.35
HTT P42858 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30224898 1.00 THRB (0.44) THRBNT5EGSK3ACDK9CDK5
SCHEMBL10220696 0.81 GSK3A (0.42) THRBNT5EGSK3ACDK9CDK5
SCHEMBL28405956 0.79 GSK3A (0.40) THRBGSK3ACDK9CDK5TAOK1
SCHEMBL30619292 0.79 GSK3A (0.40) THRBGSK3ACDK9CDK5TAOK1
SCHEMBL5660630 0.76 CYP1A2 (0.48) KDM4ETRPV4CYP2A6MAPTCYP1A2
SCHEMBL31391610 0.76 CYP1A2 (0.48) KDM4ETRPV4CYP2A6MAPTCYP1A2
SCHEMBL1519794 0.75 GSK3A (0.45) THRBGSK3ACDK9CDK5TAOK1
SCHEMBL10220699 0.74 CYP2A6 (0.42) THRBGSK3ACDK9CDK5TAOK1
SCHEMBL2117037 0.72 NT5E (0.57) THRBNT5EKDM4ECYP2A6MEN1
SCHEMBL133375 0.71 TRPV4 (0.58) NT5EKDM4ETRPV4ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-115698009-A CD73 inhibiting 2,4-dioxopyrimidine compounds 吉利德科学公司 2023-02-03 CN disclosed