SCHEMBL28952452

SCHEMBL28952452

COC(=O)c1ccc(-c2cc(-c3nc(Br)cnc3NC(=O)OC(C)(C)C)on2)cc1

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PKM P14618 1/20 0.40
MAPT P10636 5/20 0.40
NPC1 O15118 4/20 0.40
RAB9A P51151 4/20 0.40
ALDH1A1 P00352 2/20 0.40
HDAC1 Q13547 6/20 0.40
HDAC6 Q9UBN7 5/20 0.40
TP53 P04637 2/20 0.39
ATM Q13315 1/20 0.39
HDAC3 O15379 4/20 0.39
HDAC10 Q969S8 3/20 0.39
HDAC2 Q92769 3/20 0.38
HDAC8 Q9BY41 3/20 0.38
PPARA Q07869 1/20 0.37
LCK P06239 1/20 0.37
CHRM1 P11229 1/20 0.37
HDAC4 P56524 1/20 0.35
HDAC7 Q8WUI4 1/20 0.35
HDAC11 Q96DB2 1/20 0.35
HDAC9 Q9UKV0 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL25042948 0.84 ATR (0.53) ATMATR
SCHEMBL30275259 0.84 ATR (0.53) ATMATR
SCHEMBL30829221 0.82 PKM (0.40) PKMMAPTNPC1RAB9AALDH1A1
SCHEMBL29244004 0.82 PKM (0.40) PKMMAPTNPC1RAB9AALDH1A1
SCHEMBL25042592 0.81 ATR (0.48) MAPTNPC1RAB9AALDH1A1TP53
SCHEMBL28952341 0.80 HDAC1 (0.35) HDAC1HDAC6HDAC3HDAC10HDAC2
SCHEMBL14866975 0.78 ATR (0.39) HDAC1HDAC6ATMHDAC3HDAC10
SCHEMBL25042568 0.77 ATR (0.55) ATMATR
SCHEMBL13178629 0.74 GLS (0.33) HDAC1HDAC6HDAC3HDAC10HDAC2
SCHEMBL13178677 0.74 ATR (0.55) ATMATR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-115703768-A Compounds useful as inhibitors of ATR kinase 苏州爱科百发生物医药技术有限公司 2023-02-17 CN disclosed