SCHEMBL28953735

SCHEMBL28953735

COc1ccc(CSc2cc(-c3ccccc3-n3nc(C)cc3-c3ccccc3)ccc2N)cc1

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CKS1B P61024 5/20 0.41
SKP2 Q13309 5/20 0.41
NPC1 O15118 4/20 0.40
RAB9A P51151 4/20 0.40
ALDH1A1 P00352 4/20 0.40
TSHR P16473 1/20 0.40
MAPK1 P28482 3/20 0.38
SMN1; SMN2 Q16637 3/20 0.38
HPGD P15428 2/20 0.38
GAA P10253 1/20 0.38
MEN1 O00255 2/20 0.38
KMT2A Q03164 2/20 0.38
KDM4E B2RXH2 2/20 0.38
MAPT P10636 3/20 0.38
STAT1 P42224 2/20 0.38
TDP1 Q9NUW8 1/20 0.38
LMNA P02545 3/20 0.37
PDE6D O43924 1/20 0.37
PLAU P00749 1/20 0.37
FABP3 P05413 2/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28299743 0.81 RAB9A (0.53) NPC1RAB9AALDH1A1MAPK1SMN1; SMN2
SCHEMBL28847575 0.79 CSF1R (0.43) NPC1RAB9AALDH1A1TSHRMAPK1
SCHEMBL16536466 0.78 POLB (0.47) NPC1RAB9AALDH1A1TSHRSMN1; SMN2
SCHEMBL28299561 0.74 NPC1 (0.49) NPC1RAB9AALDH1A1MAPK1SMN1; SMN2
SCHEMBL28299729 0.73 NPC1 (0.46) NPC1RAB9AALDH1A1MAPK1SMN1; SMN2
SCHEMBL28301083 0.73 CA1 (0.46) NPC1RAB9AALDH1A1MAPK1SMN1; SMN2
SCHEMBL28300981 0.73 CCKAR (0.45) RAB9AFABP3FABP4
SCHEMBL28299787 0.72 NPC1 (0.47) NPC1RAB9AALDH1A1MAPK1HPGD
SCHEMBL28301021 0.72 CA1 (0.55) RAB9AFABP3FABP4
SCHEMBL19926970 0.70 NPC1 (0.45) NPC1RAB9AALDH1A1MAPK1SMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-109890822-B Inhibitors of cellular metabolic processes 安吉奥斯医药品有限公司 2022-08-30 CN disclosed