SCHEMBL28960554

SCHEMBL28960554

COCCOc1ccc(Nc2ncc(F)c(Nc3cccc(NCc4ccc(C(=O)NO)cc4)c3)n2)cc1

nearest known ligand 0.66

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
EGFR P00533 12/20 0.66
BTK Q06187 6/20 0.66
ITK Q08881 4/20 0.66
JAK3 P52333 2/20 0.66
JAK2 O60674 1/20 0.66
LYN P07948 1/20 0.66
TEC P42680 1/20 0.66
TXK P42681 1/20 0.66
BMX P51813 1/20 0.66
CD69 Q07108 1/20 0.66
SYK P43405 4/20 0.60
CCNT1 O60563 1/20 0.56
CCNE1 P24864 1/20 0.56
CDK2 P24941 1/20 0.56
CDK9 P50750 1/20 0.56

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28908376 0.89 EGFR (0.62) EGFRBTKITKJAK3JAK2
SCHEMBL30843981 0.88 EGFR (0.72) EGFRBTKITKJAK3JAK2
SCHEMBL28711237 0.88 EGFR (0.72) EGFRBTKITKJAK3JAK2
SCHEMBL28720308 0.88 EGFR (0.65) EGFRBTKITKJAK3JAK2
Benzohydroxamate SCHEMBL29172335 0.85 EGFR (0.62) EGFRBTKITKJAK3JAK2
SCHEMBL30726866 0.84 EGFR (0.68) EGFRBTKITKJAK3JAK2
SCHEMBL28908383 0.84 EGFR (0.68) EGFRBTKITKJAK3JAK2
SCHEMBL30726867 0.83 EGFR (0.67) EGFRBTKITKJAK3JAK2
SCHEMBL28908362 0.83 EGFR (0.67) EGFRBTKITKJAK3JAK2
SCHEMBL12518393 0.82 EGFR (0.73) EGFRBTKITKJAK3JAK2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-115286583-A Diphenylaminopyrimidine-containing compound, preparation and application thereof as HDACs enzyme inhibitor 山东大学 2022-11-04 CN claimed
CN-115286583-B Diphenylamino pyrimidine-containing compound, preparation and application thereof as HDACs enzyme inhibitor 山东大学 2024-01-30 CN disclosed
CN-115286583-A Diphenylaminopyrimidine-containing compound, preparation and application thereof as HDACs enzyme inhibitor 山东大学 2022-11-04 CN disclosed