SCHEMBL28720308

SCHEMBL28720308

COCCOc1ccc(Nc2ncc(F)c(Nc3ccc(C(=O)NO)cc3)n2)cc1

nearest known ligand 0.65

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
EGFR P00533 8/20 0.65
BTK Q06187 3/20 0.65
ITK Q08881 3/20 0.65
JAK2 O60674 2/20 0.65
JAK3 P52333 2/20 0.65
LYN P07948 1/20 0.65
TEC P42680 1/20 0.65
TXK P42681 1/20 0.65
BMX P51813 1/20 0.65
CD69 Q07108 1/20 0.65
SYK P43405 6/20 0.65
AURKA O14965 5/20 0.63
BRD4 O60885 1/20 0.59
RET P07949 1/20 0.59
JAK1 P23458 1/20 0.59
TYK2 P29597 1/20 0.59
FLT3 P36888 1/20 0.59
HDAC1 Q13547 1/20 0.59
HDAC8 Q9BY41 1/20 0.59
HDAC6 Q9UBN7 1/20 0.59

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28704339 0.92 EGFR (0.65) EGFRBTKITKJAK2JAK3
SCHEMBL29411908 0.92 EGFR (0.65) EGFRBTKITKJAK2JAK3
SCHEMBL28704792 0.91 EGFR (0.66) EGFRBTKITKJAK2JAK3
SCHEMBL29411905 0.91 EGFR (0.66) EGFRBTKITKJAK2JAK3
SCHEMBL28711237 0.90 EGFR (0.72) EGFRBTKITKJAK2JAK3
SCHEMBL30843981 0.90 EGFR (0.72) EGFRBTKITKJAK2JAK3
SCHEMBL28960554 0.88 EGFR (0.66) EGFRBTKITKJAK2JAK3
SCHEMBL28716958 0.85 EGFR (0.61) EGFRBTKITKJAK2JAK3
SCHEMBL23408964 0.85 SYK (0.68) EGFRBTKITKJAK2JAK3
SCHEMBL22909543 0.85 SYK (0.69) EGFRBTKITKJAK2JAK3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-114181161-B (2- ((substituted oxy) phenyl) amino) pyrimidin-4-yl) aminobenzoyl derivative and preparation method and application thereof 南通大学 2024-02-27 CN claimed
CN-114181161-A (2- ((substituted oxy) phenyl) amino) pyrimidine-4-yl) aminobenzoyl derivative and preparation method and application thereof 南通大学 2022-03-15 CN claimed
CN-114181161-B (2- ((substituted oxy) phenyl) amino) pyrimidin-4-yl) aminobenzoyl derivative and preparation method and application thereof 南通大学 2024-02-27 CN disclosed
CN-114181161-A (2- ((substituted oxy) phenyl) amino) pyrimidine-4-yl) aminobenzoyl derivative and preparation method and application thereof 南通大学 2022-03-15 CN disclosed