SCHEMBL2896243

SCHEMBL2896243

Cc1cc(Cl)cc(C(=O)N(Cc2ccccc2)C2(C)CNC2)c1C(N)=O

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KLK1 P06870 3/20 0.39
HSP90AA1 P07900 1/20 0.35
TMEM97 Q5BJF2 2/20 0.35
SIGMAR1 Q99720 2/20 0.35
MITF O75030 1/20 0.35
RAD52 P43351 1/20 0.35
KMT2A Q03164 2/20 0.34
MEN1 O00255 1/20 0.34
PDK1 Q15118 1/20 0.34
ADRA1D P25100 1/20 0.33
KDM4E B2RXH2 1/20 0.33
ALDH1A1 P00352 1/20 0.33
HPGD P15428 1/20 0.33
SMN1; SMN2 Q16637 1/20 0.33
TSHR P16473 1/20 0.33
MAPK1 P28482 1/20 0.33
LMNA P02545 1/20 0.33
NPC1 O15118 1/20 0.33
RAB9A P51151 1/20 0.33
MRGPRX4 Q96LA9 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2896247 0.88 HSP90AA1 (0.37) KLK1HSP90AA1TMEM97SIGMAR1MITF
SCHEMBL2896244 0.68 GAA (0.39) KMT2AMEN1ADRA1DKDM4EALDH1A1
SCHEMBL2783257 0.64 TSHR (0.48) KMT2AMEN1KDM4EALDH1A1TSHR
SCHEMBL5592055 0.64 NPSR1 (0.41) LMNANPC1RAB9A
SCHEMBL4666210 0.63 POLB (0.45) KMT2AKDM4EALDH1A1HPGDSMN1; SMN2
SCHEMBL14697652 0.62 ALDH1A1 (0.42) KMT2AMEN1KDM4EALDH1A1HPGD
SCHEMBL4639194 0.62 POLB (0.59) KMT2AMEN1KDM4EALDH1A1HPGD
SCHEMBL14697609 0.62 POLB (0.36) KDM4EALDH1A1HPGDSMN1; SMN2TSHR
SCHEMBL3922931 0.61 POLB (0.53) KMT2AMEN1ALDH1A1HPGDSMN1; SMN2
SCHEMBL11689298 0.61 HSP90AA1 (0.60) HSP90AA1KMT2AMEN1KDM4EALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8278464-B2 Insecticides SYNGENTA CROP PROTECTION LLC (US) 2012-10-02 US disclosed
US-8084474-B2 Insecticides SYNGENTA CROP PROTECTION, INC. (US) 2011-12-27 US disclosed
EP-2213167-A1 Anthranilamide derivatives and their use for the control of insects and acari Syngenta Participations AG (CH) 2010-08-04 EP disclosed
US-20100168066-A1 NOVEL INSECTICIDES SYNGENTA CROP PROTECTION, INC. (US) 2010-07-01 US disclosed
EP-1976385-A2 ANTHRANILAMIDE DERIVATIVES AND THEIR USE FOR THE CONTROL OF INSECTS AND ACARI Syngeta Participations AG (CH) 2008-10-08 EP disclosed
WO-2007080131-A2 ANTHRANILAMIDE DERIVATIVES AND THEIR USE FOR THE CONTROL OF INSECTS AND ACARI SYNGENTA PARTICIPATIONS AG (CH) 2007-07-19 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20100168066-A1 NOVEL INSECTICIDES DDT, ACHE, CYP4F11 KLK1 4323/4885HSP90AA1 2988/4885TMEM97 4562/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.