SCHEMBL28974406

SCHEMBL28974406

COCCN1CCN(c2ccc(C[C@H](NC(=O)OC(C)(C)C)C(=O)Nc3ccc(C(=O)O)cc3)cc2)C(=O)C1

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HDAC8 Q9BY41 1/20 0.44
AKT1 P31749 1/20 0.40
HRH2 P25021 1/20 0.40
HRH1 P35367 1/20 0.40
ITGB3 P05106 1/20 0.40
ITGB1 P05556 1/20 0.40
ITGAV P06756 1/20 0.40
ITGA2B P08514 1/20 0.40
ITGB5 P18084 1/20 0.40
CTSS P25774 6/20 0.39
CTSK P43235 5/20 0.39
CTSL P07711 2/20 0.39
CMA1 P23946 1/20 0.38
PTPN1 P18031 2/20 0.38
SCN9A Q15858 3/20 0.38
CCKAR P32238 1/20 0.38
CCKBR P32239 1/20 0.38
CTSB P07858 1/20 0.38
L3MBTL1 Q9Y468 1/20 0.38
ITGA4 P13612 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28974412 1.00 HDAC8 (0.44) HDAC8AKT1HRH2HRH1ITGB3
SCHEMBL29139621 0.94 HDAC8 (0.42) HDAC8AKT1HRH2HRH1ITGB3
SCHEMBL23486345 0.94 HDAC8 (0.42) HDAC8AKT1HRH2HRH1ITGB3
SCHEMBL28974559 0.91 HDAC8 (0.46) HDAC8AKT1HRH2HRH1ITGB3
SCHEMBL28974568 0.91 HDAC8 (0.46) HDAC8AKT1HRH2HRH1ITGB3
SCHEMBL28974608 0.89 L3MBTL1 (0.49) HDAC8AKT1ITGB3ITGB1ITGAV
SCHEMBL28974603 0.89 L3MBTL1 (0.49) HDAC8AKT1ITGB3ITGB1ITGAV
SCHEMBL28974567 0.88 HDAC8 (0.44) HDAC8AKT1ITGB3ITGB1ITGAV
SCHEMBL28974565 0.88 HDAC8 (0.44) HDAC8AKT1ITGB3ITGB1ITGAV
SCHEMBL28974517 0.88 HDAC8 (0.44) HDAC8HRH2HRH1CTSSCTSK

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-114728917-B Oxamide derivative, preparation method and medical application thereof 深圳信立泰药业股份有限公司 2023-12-08 CN disclosed
CN-114728917-A Oxamide derivative, preparation method and medical application thereof 深圳信立泰药业股份有限公司 2022-07-08 CN disclosed